{"id":29068,"date":"2019-08-08T05:30:40","date_gmt":"2019-08-08T03:30:40","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=29068"},"modified":"2019-08-08T05:30:40","modified_gmt":"2019-08-08T03:30:40","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-el-acido-ursolico-inhibe-la-proliferacion-e-induce-apoptosis-al-inactivar-la-senalizacion-de-wnt-%ce%b2-catenina-en-celulas-d","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=29068","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abEl \u00e1cido urs\u00f3lico inhibe la proliferaci\u00f3n e induce apoptosis al inactivar la se\u00f1alizaci\u00f3n de Wnt \/ \u03b2-catenina en c\u00e9lulas de osteosarcoma humano\u00bb"},"content":{"rendered":"\n<div class=\"wp-block-image\"><figure class=\"alignleft\"><a href=\"https:\/\/1.bp.blogspot.com\/-aTvVsJtUc5A\/XUsdnBXDKUI\/AAAAAAAAWMw\/aMRN4_aKL2QydWakF3EmP_nLLsGFinBLQCLcBGAs\/s1600\/International_Journal%2Bof%2BOncology.jpg\"><img decoding=\"async\" src=\"https:\/\/1.bp.blogspot.com\/-aTvVsJtUc5A\/XUsdnBXDKUI\/AAAAAAAAWMw\/aMRN4_aKL2QydWakF3EmP_nLLsGFinBLQCLcBGAs\/s1600\/International_Journal%2Bof%2BOncology.jpg\" alt=\"\"\/><\/a><\/figure><\/div>\n\n\n\n<p>Zhang, R. X., Li, Y., Tian, D. D., Liu, Y., Nian, W., Zou, X., &#8230; &amp; He, B. C. (2016).&nbsp;<a href=\"https:\/\/www.spandidos-publications.com\/10.3892\/ijo.2016.3701\">Ursolic acid inhibits proliferation and induces apoptosis by inactivating Wnt\/\u03b2-catenin signaling in human osteosarcoma cells<\/a>.&nbsp;<em>International journal of oncology<\/em>, 49(5), 1973-1982<\/p>\n\n\n\n<p>FONDO: Aunque se han utilizado m\u00faltiples agentes quimioterap\u00e9uticos para el tratamiento del osteosarcoma (OS), sus mecanismos necesitan m\u00e1s estudio. El \u00e1cido urs\u00f3lico (UA), un triterpenoide pentac\u00edclico, puede reducir la proliferaci\u00f3n celular e inducir apoptosis en varias c\u00e9lulas cancerosas, como la SG. Sin embargo, el mecanismo exacto subyacente a esta funci\u00f3n sigue sin estar claro.&nbsp;<\/p>\n\n\n\n<p>OBJETIVO: En este estudio, investigamos el efecto antiproliferativo de UA en las c\u00e9lulas OS 143B humanas y diseccionamos el posible mecanismo molecular subyacente a este efecto.&nbsp;<\/p>\n\n\n\n<p>METODO \/ DISE\u00d1O: Demostramos que la UA puede reducir la proliferaci\u00f3n celular, inducir apoptosis y detener el ciclo celular en c\u00e9lulas 143B, as\u00ed como inhibir el crecimiento tumoral de OS en un modelo de xenoinjerto de rat\u00f3n.&nbsp;<\/p>\n\n\n\n<p>RESULTADOS: Usando un ensayo de indicador de luciferasa, encontramos que la se\u00f1alizaci\u00f3n de Wnt \/ \u03b2-catenina es inhibida por UA en las c\u00e9lulas 143B. Correspondientemente, el nivel de expresi\u00f3n y la translocaci\u00f3n nuclear de \u03b2-catenina se reducen por UA. La expresi\u00f3n ex\u00f3gena de \u03b2-catenina aten\u00faa el efecto anticancer\u00edgeno de UA en las c\u00e9lulas 143B, mientras que la eliminaci\u00f3n de \u03b2-catenina aumenta este efecto. UA aumenta el nivel de expresi\u00f3n de p53 de manera dependiente de la concentraci\u00f3n, y la inhibici\u00f3n de p53 reduce el efecto anticancer\u00edgeno de UA en las c\u00e9lulas 143B. Adem\u00e1s, la inhibici\u00f3n de p53 revierte en parte la regulaci\u00f3n negativa inducida por UA de \u03b2-catenina, al igual que los objetivos de la se\u00f1alizaci\u00f3n de Wnt \/ \u03b2-catenina, como c-Myc y ciclina D1.&nbsp;<\/p>\n\n\n\n<p>CONCLUSIONES: Nuestros hallazgos indicaron que UA puede inhibir la proliferaci\u00f3n de c\u00e9lulas 143B OS a trav\u00e9s de la inactivaci\u00f3n de la se\u00f1alizaci\u00f3n de Wnt \/ \u03b2-catenina, que puede estar mediada en parte por la regulaci\u00f3n positiva de la expresi\u00f3n de p53. mientras que la eliminaci\u00f3n de \u03b2-catenina mejora este efecto.\n\n<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Zhang, R. X., Li, Y., Tian, D. D., Liu, Y., Nian, W., Zou, X., &#8230; &amp; He, B. C. (2016).&nbsp;Ursolic acid inhibits proliferation and induces apoptosis by inactivating Wnt\/\u03b2-catenin signaling in human osteosarcoma cells.&nbsp;International journal of oncology, 49(5), 1973-1982 FONDO: Aunque se han utilizado m\u00faltiples agentes quimioterap\u00e9uticos para el tratamiento del osteosarcoma (OS), sus mecanismos [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-29068","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El \u00e1cido urs\u00f3lico inhibe la proliferaci\u00f3n e induce apoptosis al inactivar la se\u00f1alizaci\u00f3n de Wnt \/ \u03b2-catenina en c\u00e9lulas de osteosarcoma humano&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=29068\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El \u00e1cido urs\u00f3lico inhibe la proliferaci\u00f3n e induce apoptosis al inactivar la se\u00f1alizaci\u00f3n de Wnt \/ \u03b2-catenina en c\u00e9lulas de osteosarcoma humano&quot; -\" \/>\n<meta property=\"og:description\" content=\"Zhang, R. X., Li, Y., Tian, D. D., Liu, Y., Nian, W., Zou, X., &#8230; &amp; He, B. C. (2016).&nbsp;Ursolic acid inhibits proliferation and induces apoptosis by inactivating Wnt\/\u03b2-catenin signaling in human osteosarcoma cells.&nbsp;International journal of oncology, 49(5), 1973-1982 FONDO: Aunque se han utilizado m\u00faltiples agentes quimioterap\u00e9uticos para el tratamiento del osteosarcoma (OS), sus mecanismos [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=29068\" \/>\n<meta property=\"article:published_time\" content=\"2019-08-08T03:30:40+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-aTvVsJtUc5A\/XUsdnBXDKUI\/AAAAAAAAWMw\/aMRN4_aKL2QydWakF3EmP_nLLsGFinBLQCLcBGAs\/s1600\/International_Journal%2Bof%2BOncology.jpg\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" 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