{"id":34796,"date":"2019-12-21T01:30:03","date_gmt":"2019-12-21T00:30:03","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=34796"},"modified":"2019-12-21T01:30:03","modified_gmt":"2019-12-21T00:30:03","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-la-apigenina-en-la-dieta-potencia-el-efecto-inhibidor-del-interferon-%ce%b1-sobre-la-viabilidad-de-las-celulas-cancerosas-media","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=34796","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa apigenina en la dieta potencia el efecto inhibidor del interfer\u00f3n \u03b1 sobre la viabilidad de las c\u00e9lulas cancerosas mediante la inhibici\u00f3n de la degradaci\u00f3n del receptor de interfer\u00f3n mediada por el proteasoma 26S\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-v8G8HnjWVa8\/XfadU23Ri4I\/AAAAAAAAZR0\/OleK6JosIXcr9qz4fsnTnK-8Q13UD7A1wCLcBGAsYHQ\/s1600\/Food_nutrition_research.jpg\"><img fetchpriority=\"high\" decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-v8G8HnjWVa8\/XfadU23Ri4I\/AAAAAAAAZR0\/OleK6JosIXcr9qz4fsnTnK-8Q13UD7A1wCLcBGAsYHQ\/s320\/Food_nutrition_research.jpg\" width=\"240\" height=\"320\" border=\"0\" data-original-width=\"400\" data-original-height=\"533\" \/><\/a>Li, S., Yang, L. J., Wang, P., He, Y. J., Huang, J. M., Liu, H. W., &#8230; &amp; Wang, F. (2016).<a href=\"https:\/\/www.tandfonline.com\/doi\/full\/10.3402\/fnr.v60.31288\">\u00a0Dietary apigenin potentiates the inhibitory effect of interferon-\u03b1 on cancer cell viability through inhibition of 26S proteasome-mediated interferon receptor degradation<\/a>.<i>\u00a0Food &amp; nutrition research<\/i>, 60(1), 31288.<\/p>\n<p>FONDO: Los interferones tipo I (IFN-\u03b1 \/ \u03b2) tienen actividades inmunorreguladoras y antiproliferativas amplias y potentes. Sin embargo, todav\u00eda se sabe si los flavonoides de la dieta exhiben sus propiedades antivirales y anticancer\u00edgenas al modular la funci\u00f3n de los IFN de tipo I.<\/p>\n<p>OBJETIVO: Este estudio tuvo como objetivo determinar el papel de la apigenina, un flavonoide vegetal de la dieta abundante en frutas y verduras comunes, sobre la inhibici\u00f3n de la viabilidad de las c\u00e9lulas cancerosas mediada por IFN.<\/p>\n<p>DISE\u00d1O: El efecto inhibitorio de la apigenina sobre el proteasoma 26S humano, un regulador negativo conocido de la se\u00f1alizaci\u00f3n de IFN tipo I, se evalu\u00f3 in vitro. El acoplamiento molecular se realiz\u00f3 para conocer la interacci\u00f3n entre la apigenina y las subunidades del proteasoma 26S. Tambi\u00e9n se investigaron los efectos de la apigenina en la v\u00eda JAK \/ STAT, la estabilidad del receptor de interfer\u00f3n mediado por el proteasoma 26S y la viabilidad de las c\u00e9lulas cancerosas.<\/p>\n<p>RESULTADOS: Se identific\u00f3 que la apigenina es un inhibidor potente del proteasoma 26S humano en un ensayo basado en c\u00e9lulas. La apigenina inhibi\u00f3 las actividades similares a la quimotripsina, a la caspasa y a la tripsina del proteasoma 26S humano y aument\u00f3 la ubiquitinaci\u00f3n de las prote\u00ednas end\u00f3genas en las c\u00e9lulas. Los resultados del modelado computacional de las posibles interacciones de apigenina con el sitio de quimotripsina (subunidad \u03b25), el sitio de caspasa (subunidad \u03b21) y el sitio de tripsina (subunidad \u03b22) del proteasoma fueron consistentes con la actividad inhibitoria del proteasoma observada. La apigenina mejor\u00f3 la fosforilaci\u00f3n del transductor de se\u00f1al y el activador de las prote\u00ednas de transcripci\u00f3n (STAT1 y STAT2) y promovi\u00f3 la expresi\u00f3n g\u00e9nica regulada por IFN-\u03b1 end\u00f3geno. La apigenina inhibi\u00f3 la ubiquitinaci\u00f3n y degradaci\u00f3n estimulada por IFN-\u03b1 del receptor 1 de interfer\u00f3n tipo I (IFNAR1).<\/p>\n<p>CONCLUSI\u00d3N: Estos resultados sugieren que la apigenina potencia el efecto inhibidor del IFN-\u03b1 sobre la viabilidad de las c\u00e9lulas cancerosas mediante la activaci\u00f3n de la v\u00eda de se\u00f1alizaci\u00f3n JAK \/ STAT a trav\u00e9s de la inhibici\u00f3n de la degradaci\u00f3n del IFNAR1 mediada por el proteasoma 26S. Esto puede proporcionar un nuevo mecanismo para aumentar la eficacia de IFN-\u03b1 \/ \u03b2.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Li, S., Yang, L. J., Wang, P., He, Y. J., Huang, J. M., Liu, H. W., &#8230; &amp; Wang, F. (2016).\u00a0Dietary apigenin potentiates the inhibitory effect of interferon-\u03b1 on cancer cell viability through inhibition of 26S proteasome-mediated interferon receptor degradation.\u00a0Food &amp; nutrition research, 60(1), 31288. FONDO: Los interferones tipo I (IFN-\u03b1 \/ \u03b2) tienen actividades [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-34796","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La apigenina en la dieta potencia el efecto inhibidor del interfer\u00f3n \u03b1 sobre la viabilidad de las c\u00e9lulas cancerosas mediante la inhibici\u00f3n de la degradaci\u00f3n del receptor de interfer\u00f3n mediada por el proteasoma 26S&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=34796\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La apigenina en la dieta potencia el efecto inhibidor del interfer\u00f3n \u03b1 sobre la viabilidad de las c\u00e9lulas cancerosas mediante la inhibici\u00f3n de la degradaci\u00f3n del receptor de interfer\u00f3n mediada por el proteasoma 26S&quot; -\" \/>\n<meta property=\"og:description\" content=\"Li, S., Yang, L. J., Wang, P., He, Y. J., Huang, J. M., Liu, H. W., &#8230; &amp; Wang, F. (2016).\u00a0Dietary apigenin potentiates the inhibitory effect of interferon-\u03b1 on cancer cell viability through inhibition of 26S proteasome-mediated interferon receptor degradation.\u00a0Food &amp; nutrition research, 60(1), 31288. FONDO: Los interferones tipo I (IFN-\u03b1 \/ \u03b2) tienen actividades [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=34796\" \/>\n<meta property=\"article:published_time\" content=\"2019-12-21T00:30:03+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-v8G8HnjWVa8\/XfadU23Ri4I\/AAAAAAAAZR0\/OleK6JosIXcr9qz4fsnTnK-8Q13UD7A1wCLcBGAsYHQ\/s320\/Food_nutrition_research.jpg\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" content=\"Tiempo de lectura\" \/>\n\t<meta name=\"twitter:data2\" content=\"2 minutos\" \/>\n<script type=\"application\/ld+json\" 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J., Wang, P., He, Y. J., Huang, J. M., Liu, H. W., &#8230; &amp; Wang, F. (2016).\u00a0Dietary apigenin potentiates the inhibitory effect of interferon-\u03b1 on cancer cell viability through inhibition of 26S proteasome-mediated interferon receptor degradation.\u00a0Food &amp; nutrition research, 60(1), 31288. FONDO: Los interferones tipo I (IFN-\u03b1 \/ \u03b2) tienen actividades [&hellip;]","og_url":"https:\/\/rina.naturopatiadigital.eu\/?p=34796","article_published_time":"2019-12-21T00:30:03+00:00","og_image":[{"url":"https:\/\/1.bp.blogspot.com\/-v8G8HnjWVa8\/XfadU23Ri4I\/AAAAAAAAZR0\/OleK6JosIXcr9qz4fsnTnK-8Q13UD7A1wCLcBGAsYHQ\/s320\/Food_nutrition_research.jpg"}],"author":"admin","twitter_card":"summary_large_image","twitter_misc":{"Escrito por":"admin","Tiempo de lectura":"2 minutos"},"schema":{"@context":"https:\/\/schema.org","@graph":[{"@type":"Article","@id":"https:\/\/rina.naturopatiadigital.eu\/?p=34796#article","isPartOf":{"@id":"https:\/\/rina.naturopatiadigital.eu\/?p=34796"},"author":{"name":"admin","@id":"https:\/\/rina.naturopatiadigital.eu\/#\/schema\/person\/432852c9ed996fc42e869a813ecbffd7"},"headline":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa apigenina en la dieta potencia el efecto inhibidor del interfer\u00f3n \u03b1 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