{"id":36100,"date":"2020-01-18T00:30:30","date_gmt":"2020-01-17T23:30:30","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=36100"},"modified":"2020-01-18T00:30:30","modified_gmt":"2020-01-17T23:30:30","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-una-posible-medicina-herbal-antitumoral-corilagin-inhibe-el-crecimiento-de-las-celulas-de-cancer-de-ovario-al-bloquear-las-vi","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=36100","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abUna posible medicina herbal antitumoral, Corilagin, inhibe el crecimiento de las c\u00e9lulas de c\u00e1ncer de ovario al bloquear las v\u00edas de se\u00f1alizaci\u00f3n de TGF-\u03b2\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-xfch26bj0Ts\/XiMhL3vHmlI\/AAAAAAAAZ_8\/WFh0tOEQFaEki4ICxxFPj2ixH6fEy9lYgCLcBGAsYHQ\/s1600\/BMC_Complementary%2Band%2BAlternative%2BMedicine.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-xfch26bj0Ts\/XiMhL3vHmlI\/AAAAAAAAZ_8\/WFh0tOEQFaEki4ICxxFPj2ixH6fEy9lYgCLcBGAsYHQ\/s1600\/BMC_Complementary%2Band%2BAlternative%2BMedicine.jpg\" border=\"0\" data-original-width=\"153\" data-original-height=\"217\" \/><\/a>Jia, L., Jin, H., Zhou, J., Chen, L., Lu, Y., Ming, Y., &amp; Yu, Y. (2013).\u00a0<a href=\"https:\/\/bmccomplementmedtherapies.biomedcentral.com\/articles\/10.1186\/1472-6882-13-33\">A potential anti-tumor herbal medicine, Corilagin, inhibits ovarian cancer cell growth through blocking the TGF-\u03b2 signaling pathways<\/a>.\u00a0<i>BMC complementary and alternative medicine<\/i>, 13(1), 33.<\/p>\n<p>FONDO: Phyllanthus niruri L. es una hierba medicinal hepatoprotectora y antiviral bien conocida. Recientemente, identificamos a Corilagin como un componente activo principal con actividad antitumoral en esta medicina herbal. Corilagin es un miembro de la familia de los taninos que se ha descubierto en muchas plantas medicinales y se ha utilizado como agente antiinflamatorio. Sin embargo, ha habido pocos informes de los efectos antitumorales de Corilagin, y su mecanismo antitumoral no se ha investigado claramente.\u00a0<\/p>\n<p>OBJETIVO: El objetivo del presente estudio es investigar las propiedades anticancer\u00edgenas de Corilagin en las c\u00e9lulas de c\u00e1ncer de ovario.<\/p>\n<p>M\u00c9TODOS Las l\u00edneas celulares de c\u00e1ncer de ovario SKOv3ip, Hey y HO-8910PM fueron tratadas con Corilagin y analizadas por el ensayo de proliferaci\u00f3n celular Sulforhodamine B (SRB), citometr\u00eda de flujo y matriz de prote\u00ednas de fase inversa (RPPA). Corilagin se administr\u00f3 por v\u00eda intraperitoneal a ratones con xenoinjertos SKOv3ip.<\/p>\n<p>RESULTADOS: Corilagin inhibi\u00f3 el crecimiento de las l\u00edneas celulares de c\u00e1ncer de ovario SKOv3ip y Hey, con valores de CI50 de menos de 30 \u03bcM, mientras mostraba baja toxicidad contra las c\u00e9lulas normales de epitelio de la superficie ov\u00e1rica, con valores de IC50 de aproximadamente 160 \u03bcM. Corilagin indujo la detenci\u00f3n del ciclo celular en la etapa G2 \/ M y una apoptosis mejorada en las c\u00e9lulas de c\u00e1ncer de ovario. Los ensayos de inmunotransferencia demostraron que Cyclin B1, Myt1, Phospho-cdc2 y Phospho-Weel estaban regulados negativamente despu\u00e9s del tratamiento con Corilagin. El crecimiento tumoral de xenoinjerto fue significativamente menor en el grupo tratado con Corilagin en comparaci\u00f3n con el grupo control no tratado ( P&lt;0.05). M\u00e1s interesante a\u00fan, Corilagin inhibi\u00f3 la secreci\u00f3n de TGF-\u03b2 en el sobrenadante de cultivo de todas las l\u00edneas celulares de c\u00e1ncer de ovario analizadas y bloque\u00f3 la estabilizaci\u00f3n de Snail inducida por TGF-\u03b2. Por el contrario, no se observ\u00f3 una reducci\u00f3n de la secreci\u00f3n de TGF-\u03b2 en las c\u00e9lulas cancerosas tratadas con el f\u00e1rmaco citot\u00f3xico Paclitaxel, lo que sugiere que Corilagin se dirige espec\u00edficamente a la secreci\u00f3n de TGF-\u03b2. Corilagin bloque\u00f3 la activaci\u00f3n de las v\u00edas can\u00f3nicas Smad y no can\u00f3nicas ERK \/ AKT.<\/p>\n<p>CONCLUSIONES: El corilagin extra\u00eddo de Phyllanthus niruri L. act\u00faa como un agente terap\u00e9utico natural y efectivo contra el crecimiento de c\u00e9lulas de c\u00e1ncer de ovario a trav\u00e9s de una acci\u00f3n dirigida contra las v\u00edas de se\u00f1alizaci\u00f3n TGF-\u03b2 \/ AKT \/ ERK \/ Smad.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Jia, L., Jin, H., Zhou, J., Chen, L., Lu, Y., Ming, Y., &amp; Yu, Y. (2013).\u00a0A potential anti-tumor herbal medicine, Corilagin, inhibits ovarian cancer cell growth through blocking the TGF-\u03b2 signaling pathways.\u00a0BMC complementary and alternative medicine, 13(1), 33. FONDO: Phyllanthus niruri L. es una hierba medicinal hepatoprotectora y antiviral bien conocida. Recientemente, identificamos a Corilagin [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-36100","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Una posible medicina herbal antitumoral, Corilagin, inhibe el crecimiento de las c\u00e9lulas de c\u00e1ncer de ovario al bloquear las v\u00edas de se\u00f1alizaci\u00f3n de TGF-\u03b2&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=36100\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Una posible medicina herbal antitumoral, Corilagin, inhibe el crecimiento de las c\u00e9lulas de c\u00e1ncer de ovario al bloquear las v\u00edas de se\u00f1alizaci\u00f3n de TGF-\u03b2&quot; -\" \/>\n<meta property=\"og:description\" content=\"Jia, L., Jin, H., Zhou, J., Chen, L., Lu, Y., Ming, Y., &amp; Yu, Y. (2013).\u00a0A potential anti-tumor herbal medicine, Corilagin, inhibits ovarian cancer cell growth through blocking the TGF-\u03b2 signaling pathways.\u00a0BMC complementary and alternative medicine, 13(1), 33. FONDO: Phyllanthus niruri L. es una hierba medicinal hepatoprotectora y antiviral bien conocida. Recientemente, identificamos a Corilagin [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=36100\" \/>\n<meta property=\"article:published_time\" content=\"2020-01-17T23:30:30+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-xfch26bj0Ts\/XiMhL3vHmlI\/AAAAAAAAZ_8\/WFh0tOEQFaEki4ICxxFPj2ixH6fEy9lYgCLcBGAsYHQ\/s1600\/BMC_Complementary%2Band%2BAlternative%2BMedicine.jpg\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" content=\"Tiempo de lectura\" \/>\n\t<meta name=\"twitter:data2\" content=\"2 minutos\" \/>\n<script type=\"application\/ld+json\" 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