{"id":38005,"date":"2020-03-07T04:30:52","date_gmt":"2020-03-07T03:30:52","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=38005"},"modified":"2020-03-07T04:30:52","modified_gmt":"2020-03-07T03:30:52","slug":"38005","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=38005","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abEl resveratrol mitiga la inflamaci\u00f3n microglial mediada por lipopolisac\u00e1rido y A\u03b2 al inhibir la cascada de se\u00f1alizaci\u00f3n TLR4 \/ NF \u2010 \u03baB \/ STAT\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-OpIhnL7fbbI\/XmNqcrNOelI\/AAAAAAAAbOQ\/KAaCXi7Ps9U1u24m0B7ZyAXD-nvlJy8mACLcBGAsYHQ\/s1600\/Journal_Neurochemistry.jpg\"><img fetchpriority=\"high\" decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-OpIhnL7fbbI\/XmNqcrNOelI\/AAAAAAAAbOQ\/KAaCXi7Ps9U1u24m0B7ZyAXD-nvlJy8mACLcBGAsYHQ\/s320\/Journal_Neurochemistry.jpg\" width=\"243\" height=\"320\" border=\"0\" data-original-width=\"400\" data-original-height=\"526\" \/><\/a>Capiralla, H., Vingtdeux, V., Zhao, H., Sankowski, R., Al\u2010Abed, Y., Davies, P., &amp; Marambaud, P. (2012).\u00a0<a href=\"https:\/\/onlinelibrary.wiley.com\/doi\/full\/10.1111\/j.1471-4159.2011.07594.x\">Resveratrol mitigates lipopolysaccharide\u2010and A\u03b2\u2010mediated microglial inflammation by inhibiting the TLR4\/NF\u2010\u03baB\/STAT signaling cascade<\/a>.\u00a0<i>Journal of neurochemistry<\/i>, 120(3), 461-472.\u00a0<\/p>\n<p>CONTEXTO: La activaci\u00f3n de la microglia, los macr\u00f3fagos residentes del cerebro, alrededor de las placas amiloides es un sello distintivo clave de la enfermedad de Alzheimer (EA). La evidencia reciente en modelos de ratones indica que se requieren microglias para el proceso neurodegenerativo de AD. Los p\u00e9ptidos amiloides-\u03b2 (A\u03b2), los componentes centrales de las placas amiloides, pueden desencadenar la activaci\u00f3n microglial al interactuar con varios receptores tipo Toll (TLR), incluido TLR4.\u00a0<\/p>\n<p>OBJETIVO \/ M\u00c9TODO: En este estudio, mostramos que el resveratrol, un polifenol natural asociado con efectos antiinflamatorios y actualmente en ensayos cl\u00ednicos para la EA, evit\u00f3 la activaci\u00f3n de macr\u00f3fagos RAW 264.7 murinos y c\u00e9lulas microgliales BV-2 tratadas con el ligando TLR4, lipopolisac\u00e1rido (LPS) .\u00a0<\/p>\n<p>RESULTADOS: El resveratrol inhibi\u00f3 preferentemente el factor nuclear \u03ba-potenciador de la cadena ligera de las c\u00e9lulas B activadas (NF-\u03baB) en la activaci\u00f3n de la estimulaci\u00f3n con LPS al interferir con la fosforilaci\u00f3n de IKK y I\u03baB, un efecto que redujo de forma potente la estimulaci\u00f3n transcripcional de varios genes diana de NF-\u03baB, incluidos factor de necrosis tumoral \u2010 \u03b1 e interleucina \u2010 6. En consecuencia, la fosforilaci\u00f3n descendente del transductor de se\u00f1al y el activador de la transcripci\u00f3n (STAT) 1 y STAT3 tras la estimulaci\u00f3n con LPS tambi\u00e9n fue inhibida por el resveratrol. Encontramos que el resveratrol actu\u00f3 hacia arriba en la cascada de activaci\u00f3n al interferir con la oligomerizaci\u00f3n de TLR4 tras la estimulaci\u00f3n del receptor. El tratamiento con resveratrol tambi\u00e9n evit\u00f3 el efecto proinflamatorio del A\u03b2 fibrilar en los macr\u00f3fagos al inhibir potentemente el efecto del A\u03b2 en la fosforilaci\u00f3n de I\u03baB, la activaci\u00f3n de STAT1 y STAT3, y sobre el factor de necrosis tumoral \u2010 \u03b1 y la secreci\u00f3n de interleucina-6. Es importante destacar que el resveratrol administrado por v\u00eda oral en un modelo de rat\u00f3n de deposici\u00f3n cerebral amiloide disminuy\u00f3 la activaci\u00f3n microglial asociada con la formaci\u00f3n de placa amiloide cortical.\u00a0<\/p>\n<p>CONCLUSIONES: Juntos, este trabajo proporciona una fuerte evidencia de que el resveratrol tieneefectos antiinflamatorios in vitro e in vivo contra la activaci\u00f3n microglial desencadenada por A\u03b2. Otros estudios en sistemas de cultivo celular mostraron que el resveratrol actu\u00f3 a trav\u00e9s de un mecanismo que involucra la cascada de se\u00f1alizaci\u00f3n TLR4 \/ NF \u2010 \u03baB \/ STAT.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Capiralla, H., Vingtdeux, V., Zhao, H., Sankowski, R., Al\u2010Abed, Y., Davies, P., &amp; Marambaud, P. (2012).\u00a0Resveratrol mitigates lipopolysaccharide\u2010and A\u03b2\u2010mediated microglial inflammation by inhibiting the TLR4\/NF\u2010\u03baB\/STAT signaling cascade.\u00a0Journal of neurochemistry, 120(3), 461-472.\u00a0 CONTEXTO: La activaci\u00f3n de la microglia, los macr\u00f3fagos residentes del cerebro, alrededor de las placas amiloides es un sello distintivo clave de la enfermedad [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-38005","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El resveratrol mitiga la inflamaci\u00f3n microglial mediada por lipopolisac\u00e1rido y A\u03b2 al inhibir la cascada de se\u00f1alizaci\u00f3n TLR4 \/ NF \u2010 \u03baB \/ STAT&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=38005\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El resveratrol mitiga la inflamaci\u00f3n microglial mediada por lipopolisac\u00e1rido y A\u03b2 al inhibir la cascada de se\u00f1alizaci\u00f3n TLR4 \/ NF \u2010 \u03baB \/ STAT&quot; -\" \/>\n<meta property=\"og:description\" content=\"Capiralla, H., Vingtdeux, V., Zhao, H., Sankowski, R., Al\u2010Abed, Y., Davies, P., &amp; Marambaud, P. 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