{"id":41668,"date":"2020-06-01T03:30:16","date_gmt":"2020-06-01T01:30:16","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=41668"},"modified":"2020-06-01T03:30:16","modified_gmt":"2020-06-01T01:30:16","slug":"41668","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=41668","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abInhibe \u00e1cido urs\u00f3lico factor nuclear-kB se\u00f1alizaci\u00f3n en las c\u00e9lulas intestinales epiteliales y macr\u00f3fagos, y aten\u00faa la colitis experimental en ratones\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-vXFrBCKhzC4\/XtUU57XRd2I\/AAAAAAAAdQg\/q7rZKyiL-xwvl9Yc9e4wxhENAWVhFO9oACLcBGAsYHQ\/s1600\/Life_Sciences.jpg\"><img fetchpriority=\"high\" decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-vXFrBCKhzC4\/XtUU57XRd2I\/AAAAAAAAdQg\/q7rZKyiL-xwvl9Yc9e4wxhENAWVhFO9oACLcBGAsYHQ\/s320\/Life_Sciences.jpg\" width=\"240\" height=\"320\" border=\"0\" data-original-width=\"576\" data-original-height=\"768\" \/><\/a>Chun, J., Lee, C., Hwang, S. W., Im, J. P., &amp; Kim, J. S. (2014).\u00a0<a href=\"https:\/\/www.sciencedirect.com\/science\/article\/abs\/pii\/S0024320514005724\">Ursolic acid inhibits nuclear factor-\u03baB signaling in intestinal epithelial cells and macrophages, and attenuates experimental colitis in mice<\/a>.\u00a0<i>Life sciences<\/i>, 110(1), 23-34.<\/p>\n<p>OBJETIVOS: Se ha informado que el \u00e1cido urs\u00f3lico (UA), un \u00e1cido triterpenoide pentac\u00edclico natural, muestra actividad inmunomoduladora. Este estudio investig\u00f3 los efectos de la UA sobre la se\u00f1alizaci\u00f3n del factor nuclear kappa B (NF-\u03baB) en las c\u00e9lulas y la colitis murina experimental.<\/p>\n<p>M\u00c9TODOS PRINICPALES: Las c\u00e9lulas epiteliales intestinales humanas (IEC) COLO 205 y los macr\u00f3fagos peritoneales de ratones con deficiencia de IL-10 (IL-10 &#8211; \/ &#8211; ) fueron pretratados con UA \u200b\u200by luego estimulados con factor de necrosis tumoral \u03b1 (TNF-\u03b1) y lipopolisac\u00e1rido (LPS) , respectivamente. La expresi\u00f3n de citocinas proinflamatorias se determin\u00f3 mediante RT-PCR en tiempo real y ELISA. El efecto de UA sobre la se\u00f1alizaci\u00f3n de NF-\u03baB se examin\u00f3 mediante an\u00e1lisis de inmunotransferencia para detectar la fosforilaci\u00f3n \/ degradaci\u00f3n de I\u03baB\u03b1 y el ensayo de cambio de movilidad electrofor\u00e9tica para evaluar la actividad de uni\u00f3n al ADN de NF-\u03baB. Para estudios in vivo , colitis aguda inducida por sulfato s\u00f3dico de dextrano (DSS) en ratones de tipo salvaje C57BL \/ 6 y colitis cr\u00f3nica en IL-10 &#8211; \/ -los ratones fueron tratados con o sin UA. La colitis se cuantific\u00f3 por evaluaci\u00f3n histopatol\u00f3gica. La tinci\u00f3n inmunohistoqu\u00edmica para I\u03baB\u03b1 fosforilada se realiz\u00f3 en el tejido col\u00f3nico.<\/p>\n<p>RESULTADOS CLAVES: UA inhibi\u00f3 significativamente la producci\u00f3n de citocinas proinflamatorias, fosforilaci\u00f3n \/ degradaci\u00f3n de I\u03baB\u03b1 y actividad de uni\u00f3n a ADN de NF-\u03baB en macr\u00f3fagos peritoneales IEC e IL-10 &#8211; \/ &#8211; estimulados con TNF-\u03b1 y LPS, respectivamente. UA redujo significativamente la gravedad de la colitis murina inducida por DSS, seg\u00fan lo evaluado por el \u00edndice de actividad de la enfermedad, la longitud del colon y la histopatolog\u00eda. UA tambi\u00e9n mejor\u00f3 significativamente la gravedad de la colitis en ratones IL-10 &#8211; \/ &#8211; . Adem\u00e1s, UA suprimi\u00f3 la fosforilaci\u00f3n de I\u03baB\u03b1 en el tejido col\u00f3nico.<\/p>\n<p>SIGNIFICADO: UA inhibe la activaci\u00f3n de NF-\u03baB tanto en IEC como en macr\u00f3fagos, y aten\u00faa la colitis murina experimental. Estos resultados sugieren que la UA es un agente terap\u00e9utico potencial para la enfermedad inflamatoria intestinal.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Chun, J., Lee, C., Hwang, S. W., Im, J. P., &amp; Kim, J. S. (2014).\u00a0Ursolic acid inhibits nuclear factor-\u03baB signaling in intestinal epithelial cells and macrophages, and attenuates experimental colitis in mice.\u00a0Life sciences, 110(1), 23-34. OBJETIVOS: Se ha informado que el \u00e1cido urs\u00f3lico (UA), un \u00e1cido triterpenoide pentac\u00edclico natural, muestra actividad inmunomoduladora. Este estudio investig\u00f3 [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-41668","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Inhibe \u00e1cido urs\u00f3lico factor nuclear-kB se\u00f1alizaci\u00f3n en las c\u00e9lulas intestinales epiteliales y macr\u00f3fagos, y aten\u00faa la colitis experimental en ratones&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=41668\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Inhibe \u00e1cido urs\u00f3lico factor nuclear-kB se\u00f1alizaci\u00f3n en las c\u00e9lulas intestinales epiteliales y macr\u00f3fagos, y aten\u00faa la colitis experimental en ratones&quot; -\" \/>\n<meta property=\"og:description\" content=\"Chun, J., Lee, C., Hwang, S. W., Im, J. P., &amp; Kim, J. S. (2014).\u00a0Ursolic acid inhibits nuclear factor-\u03baB signaling in intestinal epithelial cells and macrophages, and attenuates experimental colitis in mice.\u00a0Life sciences, 110(1), 23-34. OBJETIVOS: Se ha informado que el \u00e1cido urs\u00f3lico (UA), un \u00e1cido triterpenoide pentac\u00edclico natural, muestra actividad inmunomoduladora. 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