{"id":42073,"date":"2020-06-10T00:30:52","date_gmt":"2020-06-09T22:30:52","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=42073"},"modified":"2020-06-10T00:30:52","modified_gmt":"2020-06-09T22:30:52","slug":"42073","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=42073","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abMecanismos implicados en la apoptosis inducida por resveratrol y la detenci\u00f3n del ciclo celular en el c\u00e1ncer de pr\u00f3stata: l\u00edneas celulares derivadas\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-dMxxyf7iaiE\/XuEn3K4tFBI\/AAAAAAAAdd0\/dfMeMwUgj5ESdkTqVq0o5l0fFqnJKgWQwCLcBGAsYHQ\/s1600\/Journal_andrology.png\"><img fetchpriority=\"high\" decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-dMxxyf7iaiE\/XuEn3K4tFBI\/AAAAAAAAdd0\/dfMeMwUgj5ESdkTqVq0o5l0fFqnJKgWQwCLcBGAsYHQ\/s320\/Journal_andrology.png\" width=\"245\" height=\"320\" border=\"0\" data-original-width=\"843\" data-original-height=\"1100\" \/><\/a>Benitez, D. A., Pozo\u2010Guisado, E., Alvarez\u2010Barrientos, A., Fernandez\u2010Salguero, P. M., &amp; Castell\u00f3n, E. A. (2007).\u00a0<a href=\"http:\/\/onlinelibrary.wiley.com\/doi\/10.2164\/jandrol.106.000968\/full\">Mechanisms Involved in Resveratrol\u2010Induced Apoptosis and Cell Cycle Arrest in Prostate Cancer\u2014Derived Cell Lines.<i>\u00a0<\/i><\/a><i>Journal of andrology<\/i>, 28(2), 282-293.\u00a0<\/p>\n<p>FONDO: El resveratrol es un polifenol encontrado en altas concentraciones en uvas y vino tinto con efectos anticancer\u00edgenos reportados.\u00a0<\/p>\n<p>OBJETIVO \/ M\u00c9TODO: Estudiamos el mecanismo molecular de la apoptosis inducida por resveratrol y la detenci\u00f3n de la proliferaci\u00f3n en c\u00e9lulas derivadas de pr\u00f3stata PZ-HPV-7 (l\u00ednea no tumorig\u00e9nica), LNCaP (l\u00ednea de c\u00e1ncer sensible a andr\u00f3genos) y PC-3 (l\u00ednea de c\u00e1ncer insensible a andr\u00f3genos). La apoptosis y la distribuci\u00f3n del ciclo celular se evaluaron mediante citometr\u00eda de flujo y proliferaci\u00f3n mediante ensayo de MTT y conteo directo de c\u00e9lulas. Las caspasas, bax, bcl-2, ciclinas, Cdks, p53, p21 y p27 se midieron por Western blot y las actividades de cinasa de complejos de ciclina \/ Cdk por inmunoprecipitaci\u00f3n seguido de ensayos de cinasa con sustratos apropiados.\u00a0<\/p>\n<p>RESULTADOS: El resveratrol indujo una disminuci\u00f3n en las tasas de proliferaci\u00f3n y un aumento en la apoptosis en l\u00edneas celulares cancerosas de una manera dependiente de la dosis y del tiempo. Estos efectos fueron coincidentes con la acumulaci\u00f3n celular en la fase G0 \/ G1. En LNCaP y PC-3, la apoptosis inducida por el resveratrol estuvo mediada por la activaci\u00f3n de las caspasas 9 y 3 y un cambio en la relaci\u00f3n de bax \/ bcl-2. Las expresiones de ciclina D1, E y Cdk4, as\u00ed como la actividad ciclina D1 \/ Cdk4 quinasa se redujeron por el resveratrol solo en c\u00e9lulas LNCaP. Por el contrario, la expresi\u00f3n de ciclina B y Cdk1 y la actividad de la ciclina B \/ Cdk1 quinasa disminuyeron en ambas l\u00edneas celulares en presencia de resveratrol. Sin embargo, las prote\u00ednas moduladoras p53, p21, y p27 se incrementaron con resveratrol solo en c\u00e9lulas LNCaP. Estos efectos probablemente dan como resultado la detenci\u00f3n de la proliferaci\u00f3n observada y la interrupci\u00f3n del control del ciclo celular. Adem\u00e1s, las diferencias espec\u00edficas encontradas entre LNCaP y PC-3 sugieren que el resveratrol act\u00faa a trav\u00e9s de diferentes mecanismos sobre el estado de las c\u00e9lulas receptoras de andr\u00f3genos o estr\u00f3genos.\u00a0<\/p>\n<p>OBSERVACIONES: Existen muy pocos estudios sobre la toxicidad del resveratrol in vivo. Recientemente, se ha informado que solo en altas dosis (3 g \/ Kg \/ d\u00eda), el resveratrol causa toxicidad hep\u00e1tica moderada seg\u00fan lo medido por el conjunto de ADN y la inducci\u00f3n de enzimas metabolizantes de fase II (Hebbar et al, 2005). Esta concentraci\u00f3n potencialmente t\u00f3xica est\u00e1 m\u00e1s all\u00e1 de las dosis utilizadas en este estudio. Finalmente, es importante se\u00f1alar que la comparaci\u00f3n de estos aspectos de los efectos del resveratrol, en las mismas condiciones experimentales, entre las c\u00e9lulas LNCaP y PC-3 es muy relevante considerando que estas c\u00e9lulas son representativas de las 2 etapas principales del c\u00e1ncer de pr\u00f3stata, a saber, andr\u00f3geno-sensible y tumores insensibles a los andr\u00f3genos.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Benitez, D. A., Pozo\u2010Guisado, E., Alvarez\u2010Barrientos, A., Fernandez\u2010Salguero, P. M., &amp; Castell\u00f3n, E. A. (2007).\u00a0Mechanisms Involved in Resveratrol\u2010Induced Apoptosis and Cell Cycle Arrest in Prostate Cancer\u2014Derived Cell Lines.\u00a0Journal of andrology, 28(2), 282-293.\u00a0 FONDO: El resveratrol es un polifenol encontrado en altas concentraciones en uvas y vino tinto con efectos anticancer\u00edgenos reportados.\u00a0 OBJETIVO \/ M\u00c9TODO: Estudiamos [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-42073","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Mecanismos implicados en la apoptosis inducida por resveratrol y la detenci\u00f3n del ciclo celular en el c\u00e1ncer de pr\u00f3stata: l\u00edneas celulares derivadas&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=42073\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Mecanismos implicados en la apoptosis inducida por resveratrol y la detenci\u00f3n del ciclo celular en el c\u00e1ncer de pr\u00f3stata: l\u00edneas celulares derivadas&quot; -\" \/>\n<meta property=\"og:description\" content=\"Benitez, D. 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