{"id":42079,"date":"2020-06-10T02:30:41","date_gmt":"2020-06-10T00:30:41","guid":{"rendered":"https:\/\/naturopatiadigital.eu\/?p=42079"},"modified":"2020-06-10T02:30:41","modified_gmt":"2020-06-10T00:30:41","slug":"42079","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=42079","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa apoptosis causada por el resveratrol de las c\u00e9lulas LNCaP del carcinoma de pr\u00f3stata humano est\u00e1 mediada por la modulaci\u00f3n de la v\u00eda de fosfatidilinositol 3&#8242;-quinasa \/ Akt y las prote\u00ednas de la familia Bcl-2\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-UKNnWwGYU1o\/XuErrFN0KxI\/AAAAAAAAdeE\/tAzmUVRKdK4j7q_tiY5jtJ-bmR8Hm53hQCLcBGAsYHQ\/s1600\/Molecular_Cancer%2BTherapeutics.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-UKNnWwGYU1o\/XuErrFN0KxI\/AAAAAAAAdeE\/tAzmUVRKdK4j7q_tiY5jtJ-bmR8Hm53hQCLcBGAsYHQ\/s1600\/Molecular_Cancer%2BTherapeutics.jpg\" border=\"0\" data-original-width=\"195\" data-original-height=\"259\" \/><\/a>Aziz, M. H., Nihal, M., Fu, V. X., Jarrard, D. F., &amp; Ahmad, N. (2006).\u00a0<a href=\"http:\/\/mct.aacrjournals.org\/content\/5\/5\/1335.short\">Resveratrol-caused apoptosis of human prostate carcinoma LNCaP cells is mediated via modulation of phosphatidylinositol 3\u2032-kinase\/Akt pathway and Bcl-2 family proteins<\/a>.\u00a0<i>Molecular cancer therapeutics,<\/i>\u00a05(5), 1335-1341.\u00a0<\/p>\n<p>FONDO: El c\u00e1ncer de pr\u00f3stata es un problema de salud importante en los EE. UU. Y el tratamiento disponible y las opciones quir\u00fargicas han demostrado ser insuficientes para controlar la mortalidad y la morbilidad asociadas con esta enfermedad. Por lo tanto, es necesario intensificar nuestros esfuerzos para comprender mejor esta enfermedad y desarrollar nuevos enfoques para su prevenci\u00f3n y tratamiento.\u00a0<\/p>\n<p>OBJETIVO: Este estudio se realiz\u00f3 para evaluar el potencial quimiopreventivo \/ antiproliferativo del resveratrol (trans -3,4 &#8216;, 5, -trihydroxystilbene) contra el c\u00e1ncer de pr\u00f3stata y su mecanismo de acci\u00f3n.\u00a0<\/p>\n<p>RESULTADOS: El tratamiento con resveratrol (0-50 \u03bcmol \/ L durante 24 horas) produjo unadisminuci\u00f3n significativa (a) en la viabilidad celular, (b) disminuci\u00f3n de la supervivencia de las c\u00e9lulas clonog\u00e9nicas, (c) inhibici\u00f3n del crecimiento estimulado por andr\u00f3genos (R1881), y (d) inducci\u00f3n de apoptosis en c\u00e9lulas de carcinoma de pr\u00f3stata humano (LNCaP) sensible a andr\u00f3genos. Curiosamente, a concentraciones similares, el tratamiento con resveratrol no afect\u00f3 la viabilidad o tasa de apoptosis en c\u00e9lulas epiteliales de pr\u00f3stata humanas normales. Adem\u00e1s, nuestros datos mostraron que el tratamiento con resveratrol result\u00f3 en una inhibici\u00f3n dependiente de la dosis significativa en la expresi\u00f3n constitutiva de fosfatidilinositol 3&#8242;-quinasa y Akt fosforilada (activa) en c\u00e9lulas LNCaP. Tambi\u00e9n se encontr\u00f3 que el tratamiento con resveratrol para c\u00e9lulas LNCaP resulta en una (a) p\u00e9rdida significativa del potencial de membrana mitocondrial, (b) inhibici\u00f3n en el nivel de prote\u00edna de Bcl-2 antiapopt\u00f3tico, y (c) aumento en los miembros proapopt\u00f3ticos de la familia Bcl-2, es decir, Bax, Bak, Bid y Bad.\u00a0<\/p>\n<p>CONCLUSIONES: Tomados en conjunto, nuestros datos sugieren que el resveratrol causa una inhibici\u00f3n de la activaci\u00f3n de la fosfatidilinositol 3&#8242;-quinasa \/ Akt que, a su vez, produce modulaciones en las prote\u00ednas de la familia Bcl-2 de tal manera que se promueve la apoptosis de las c\u00e9lulas LNCaP. Con base en estos estudios, sugerimos que el resveratrol podr\u00eda desarrollarse como un agente para el tratamiento del c\u00e1ncer de pr\u00f3stata.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Aziz, M. H., Nihal, M., Fu, V. X., Jarrard, D. F., &amp; Ahmad, N. (2006).\u00a0Resveratrol-caused apoptosis of human prostate carcinoma LNCaP cells is mediated via modulation of phosphatidylinositol 3\u2032-kinase\/Akt pathway and Bcl-2 family proteins.\u00a0Molecular cancer therapeutics,\u00a05(5), 1335-1341.\u00a0 FONDO: El c\u00e1ncer de pr\u00f3stata es un problema de salud importante en los EE. UU. Y el tratamiento [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-42079","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La apoptosis causada por el resveratrol de las c\u00e9lulas LNCaP del carcinoma de pr\u00f3stata humano est\u00e1 mediada por la modulaci\u00f3n de la v\u00eda de fosfatidilinositol 3&#039;-quinasa \/ Akt y las prote\u00ednas de la familia Bcl-2&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=42079\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La apoptosis causada por el resveratrol de las c\u00e9lulas LNCaP del carcinoma de pr\u00f3stata humano est\u00e1 mediada por la modulaci\u00f3n de la v\u00eda de fosfatidilinositol 3&#039;-quinasa \/ Akt y las prote\u00ednas de la familia Bcl-2&quot; -\" \/>\n<meta property=\"og:description\" content=\"Aziz, M. H., Nihal, M., Fu, V. X., Jarrard, D. F., &amp; Ahmad, N. (2006).\u00a0Resveratrol-caused apoptosis of human prostate carcinoma LNCaP cells is mediated via modulation of phosphatidylinositol 3\u2032-kinase\/Akt pathway and Bcl-2 family proteins.\u00a0Molecular cancer therapeutics,\u00a05(5), 1335-1341.\u00a0 FONDO: El c\u00e1ncer de pr\u00f3stata es un problema de salud importante en los EE. UU. Y el tratamiento [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=42079\" \/>\n<meta property=\"article:published_time\" content=\"2020-06-10T00:30:41+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-UKNnWwGYU1o\/XuErrFN0KxI\/AAAAAAAAdeE\/tAzmUVRKdK4j7q_tiY5jtJ-bmR8Hm53hQCLcBGAsYHQ\/s1600\/Molecular_Cancer%2BTherapeutics.jpg\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" content=\"Tiempo de lectura\" \/>\n\t<meta name=\"twitter:data2\" content=\"2 minutos\" \/>\n<script type=\"application\/ld+json\" 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