{"id":43935,"date":"2020-09-04T03:30:07","date_gmt":"2020-09-04T01:30:07","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=43935"},"modified":"2020-09-06T09:47:07","modified_gmt":"2020-09-06T07:47:07","slug":"43935","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=43935","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abActividad antitumoral y eventos de se\u00f1alizaci\u00f3n desencadenados por isotiocianatos, sulforafano e isotiocianato de fenetilo, en el mieloma m\u00faltiple\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-W3F98MaPIrA\/X1STdmauL-I\/AAAAAAAAfnc\/h-8XzTmobhIbP32ZAiHjb7QkyMmOr71MQCLcBGAsYHQ\/s1600\/Haematologica.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-W3F98MaPIrA\/X1STdmauL-I\/AAAAAAAAfnc\/h-8XzTmobhIbP32ZAiHjb7QkyMmOr71MQCLcBGAsYHQ\/s1600\/Haematologica.jpg\" border=\"0\" data-original-width=\"165\" data-original-height=\"220\" \/><\/a>Jakubikova, J., Cervi, D., Ooi, M., Kim, K., Nahar, S., Klippel, S., &#8230; &amp; Negri, J. (2011).\u00a0<a href=\"https:\/\/haematologica.org\/article\/view\/6044\">Anti-tumor activity and signaling events triggered by the isothiocyanates, sulforaphane and phenethyl isothiocyanate, in multiple myeloma<\/a>.\u00a0<i>Haematologica<\/i>, 96(8), 1170-1179.<\/p>\n<p>ANTECEDENTES: Los isotiocianatos, una familia de fitoqu\u00edmicos que se encuentran en las verduras cruc\u00edferas, tienen efectos citot\u00f3xicos contra varios tipos de c\u00e9lulas tumorales. El mieloma m\u00faltiple es una enfermedad mortal caracterizada por la proliferaci\u00f3n clonal de c\u00e9lulas plasm\u00e1ticas en la m\u00e9dula \u00f3sea.<\/p>\n<p>OBJETIVO: El creciente cuerpo de informaci\u00f3n precl\u00ednica sobre la actividad anticancer\u00edgena de los isotiocianatos nos llev\u00f3 a investigar sus propiedades antimieloma.<\/p>\n<p>DISE\u00d1O Y METODOS: Se evalu\u00f3 la actividad anti-mieloma de los isotiocianatos, sulforafano e isotiocianato de fenetilo, en un panel de l\u00edneas celulares de mieloma humano, as\u00ed como c\u00e9lulas tumorales de mieloma primario. La viabilidad celular, la apoptosis, las alteraciones del ciclo celular y la proliferaci\u00f3n celular se analizaron in vitro y en un modelo de rat\u00f3n de xenoinjerto in vivo.. Las secuelas moleculares del tratamiento con isotiocianato en c\u00e9lulas de mieloma m\u00faltiple se evaluaron mediante an\u00e1lisis multiplex utilizando matrices de perlas y transferencia Western.<\/p>\n<p>RESULTADOS: Observamos que el sulforafano y el isotiocianato de feniletilo tienen actividad contra las l\u00edneas celulares de mieloma y las c\u00e9lulas de mieloma de los pacientes tanto in vitro como in vivo utilizando un modelo de rat\u00f3n de xenoinjerto de mieloma. Los isotiocianatos indujeron la muerte apopt\u00f3tica de las c\u00e9lulas de mieloma; agotamiento del potencial de la membrana mitocondrial; escisi\u00f3n de PARP y caspasas-3 y -9; as\u00ed como la regulaci\u00f3n a la baja de prote\u00ednas anti-apopt\u00f3ticas que incluyen Mcl-1, X-IAP, c-IAP y survivina. G 2 inducido por isotiocianatos\/ M parada del ciclo celular acompa\u00f1ada de fosforilaci\u00f3n mit\u00f3tica de histona H3. El an\u00e1lisis multiplex de fosforilaci\u00f3n de diversos componentes de las cascadas de se\u00f1alizaci\u00f3n revel\u00f3 cambios en la activaci\u00f3n de MAPK; aumento de la fosforilaci\u00f3n de c-jun y HSP27; as\u00ed como cambios en la fosforilaci\u00f3n de Akt, GSK3\u03b1 \/ \u03b2 y p53. Los isotiocianatos suprimieron la proliferaci\u00f3n de c\u00e9lulas de mieloma solas y cuando se cultivaron conjuntamente con c\u00e9lulas estromales HS-5. El sulforafano y el isotiocianato de feniletilo mejoraron la actividad anti-mieloma in vitro de varias terapias convencionales y nuevas utilizadas en el mieloma m\u00faltiple.<\/p>\n<p>CONCLUSIONES: Nuestro estudio muestra que los isotiocianatos tienen potentes actividades anti-mieloma y pueden mejorar la actividad de otros agentes anti-mieloma m\u00faltiple. Estos resultados indican que los isotiocianatos pueden tener potencial terap\u00e9utico en el mieloma m\u00faltiple y proporcionan el marco precl\u00ednico para futuros estudios cl\u00ednicos de isotiocianatos en el mieloma m\u00faltiple.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Jakubikova, J., Cervi, D., Ooi, M., Kim, K., Nahar, S., Klippel, S., &#8230; &amp; Negri, J. (2011).\u00a0Anti-tumor activity and signaling events triggered by the isothiocyanates, sulforaphane and phenethyl isothiocyanate, in multiple myeloma.\u00a0Haematologica, 96(8), 1170-1179. ANTECEDENTES: Los isotiocianatos, una familia de fitoqu\u00edmicos que se encuentran en las verduras cruc\u00edferas, tienen efectos citot\u00f3xicos contra varios tipos de [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-43935","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Actividad antitumoral y eventos de se\u00f1alizaci\u00f3n desencadenados por isotiocianatos, sulforafano e isotiocianato de fenetilo, en el mieloma m\u00faltiple&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=43935\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Actividad antitumoral y eventos de se\u00f1alizaci\u00f3n desencadenados por isotiocianatos, sulforafano e isotiocianato de fenetilo, en el mieloma m\u00faltiple&quot; -\" \/>\n<meta property=\"og:description\" content=\"Jakubikova, J., Cervi, D., Ooi, M., Kim, K., Nahar, S., Klippel, S., &#8230; &amp; Negri, J. (2011).\u00a0Anti-tumor activity and signaling events triggered by the isothiocyanates, sulforaphane and phenethyl isothiocyanate, in multiple myeloma.\u00a0Haematologica, 96(8), 1170-1179. 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