{"id":43952,"date":"2020-09-05T01:30:15","date_gmt":"2020-09-04T23:30:15","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=43952"},"modified":"2020-09-06T10:51:54","modified_gmt":"2020-09-06T08:51:54","slug":"43952","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=43952","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa ingesti\u00f3n de quercetina inhibe la agregaci\u00f3n plaquetaria y los componentes esenciales de la v\u00eda de activaci\u00f3n plaquetaria estimulada por col\u00e1geno en humanos\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-pOLzztfvCYU\/X1SitCNHRhI\/AAAAAAAAfoM\/Qm1xF5lR2ssjMk2ZmDVAYPp8NcTeMfngwCLcBGAsYHQ\/s1600\/Journal_Thrombosis%2Band%2BHaemostasis.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-pOLzztfvCYU\/X1SitCNHRhI\/AAAAAAAAfoM\/Qm1xF5lR2ssjMk2ZmDVAYPp8NcTeMfngwCLcBGAsYHQ\/s1600\/Journal_Thrombosis%2Band%2BHaemostasis.jpg\" border=\"0\" data-original-width=\"195\" data-original-height=\"258\" \/><\/a>Hubbard, G. P., Wolffram, S., Lovegrove, J. A., &amp; Gibbins, J. M. (2004).\u00a0<a href=\"https:\/\/onlinelibrary.wiley.com\/doi\/pdf\/10.1111\/j.1538-7836.2004.01067.x\">Ingestion of quercetin inhibits platelet aggregation and essential components of the collagen\u2010stimulated platelet activation pathway in humans<\/a>.\u00a0<i>Journal of Thrombosis and Haemostasis<\/i>, 2(12), 2138-2145.<\/p>\n<p>ANTECEDENTES: La quercetina, un flavonoide presente en la dieta humana, que se encuentra en niveles elevados en cebollas, manzanas, t\u00e9 y vino, ha demostrado previamente que inhibe la agregaci\u00f3n plaquetaria y la se\u00f1alizaci\u00f3n in vitro. En consecuencia, se ha propuesto que la quercetina puede contribuir a los efectos protectores frente a las enfermedades cardiovasculares de una dieta rica en frutas y verduras.<\/p>\n<p>OBJETIVOS: Se dise\u00f1\u00f3 un estudio piloto de intervenci\u00f3n diet\u00e9tica humana para investigar la relaci\u00f3n entre la ingesti\u00f3n de quercetina diet\u00e9tica y la funci\u00f3n plaquetaria.<\/p>\n<p>METODOS: Los sujetos humanos ingirieron 150 mg o 300 mg de suplemento de quercetina-4&#8242;-O-beta-D-gluc\u00f3sido para determinar la disponibilidad sist\u00e9mica de quercetina. Se aislaron plaquetas de sujetos para analizar la se\u00f1alizaci\u00f3n y agregaci\u00f3n de c\u00e9lulas estimuladas por col\u00e1geno.<\/p>\n<p>RESULTADOS: las concentraciones plasm\u00e1ticas de quercetina alcanzaron un m\u00e1ximo de 4,66 micras (+\/- 0,77) y 9,72 micras (+\/- 1,38) 30 minutos despu\u00e9s de la ingesti\u00f3n de dosis de 150 mg y 300 mg de quercetina-4&#8242;-O-beta-D-gluc\u00f3sido , respectivamente, demostrando que la quercetina estaba biodisponible, con concentraciones plasm\u00e1ticas alcanzadas en el rango conocido por afectar la funci\u00f3n plaquetaria in vitro. La agregaci\u00f3n plaquetaria se inhibi\u00f3 30 y 120 minutos despu\u00e9s de la ingesti\u00f3n de ambas dosis de quercetina-4&#8242;-O-beta-D-gluc\u00f3sido. De forma correspondiente, se inhibi\u00f3 la fosforilaci\u00f3n de tirosina estimulada por col\u00e1geno de las prote\u00ednas plaquetarias totales. Esto se acompa\u00f1\u00f3 de una reducci\u00f3n de la fosforilaci\u00f3n de tirosina de la tirosina quinasa Syk y la fosfolipasa Cgamma2, componentes de la v\u00eda de se\u00f1alizaci\u00f3n del receptor de col\u00e1geno de la glucoprote\u00edna VI plaquetaria.<\/p>\n<p>CONCLUSIONES: Este estudio proporciona nueva evidencia de la disponibilidad sist\u00e9mica relativamente alta de quercetina en forma de quercetina-4&#8242;-O-beta-D-gluc\u00f3sido mediante suplementaci\u00f3n, e implica a la quercetina como un inhibidor diet\u00e9tico de la se\u00f1alizaci\u00f3n de las c\u00e9lulas plaquetarias y la formaci\u00f3n de trombos.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Hubbard, G. P., Wolffram, S., Lovegrove, J. A., &amp; Gibbins, J. M. (2004).\u00a0Ingestion of quercetin inhibits platelet aggregation and essential components of the collagen\u2010stimulated platelet activation pathway in humans.\u00a0Journal of Thrombosis and Haemostasis, 2(12), 2138-2145. ANTECEDENTES: La quercetina, un flavonoide presente en la dieta humana, que se encuentra en niveles elevados en cebollas, manzanas, t\u00e9 [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-43952","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La ingesti\u00f3n de quercetina inhibe la agregaci\u00f3n plaquetaria y los componentes esenciales de la v\u00eda de activaci\u00f3n plaquetaria estimulada por col\u00e1geno en humanos&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=43952\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La ingesti\u00f3n de quercetina inhibe la agregaci\u00f3n plaquetaria y los componentes esenciales de la v\u00eda de activaci\u00f3n plaquetaria estimulada por col\u00e1geno en humanos&quot; -\" \/>\n<meta property=\"og:description\" content=\"Hubbard, G. P., Wolffram, S., Lovegrove, J. A., &amp; Gibbins, J. M. (2004).\u00a0Ingestion of quercetin inhibits platelet aggregation and essential components of the collagen\u2010stimulated platelet activation pathway in humans.\u00a0Journal of Thrombosis and Haemostasis, 2(12), 2138-2145. 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