{"id":44092,"date":"2020-09-18T00:30:22","date_gmt":"2020-09-17T22:30:22","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=44092"},"modified":"2020-10-02T22:22:36","modified_gmt":"2020-10-02T20:22:36","slug":"44092","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=44092","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa capsaicina suprime la migraci\u00f3n de las c\u00e9lulas del colangiocarcinoma al regular negativamente la expresi\u00f3n de la metaloproteinasa-9 de la matriz a trav\u00e9s de la v\u00eda de se\u00f1alizaci\u00f3n AMPK-NF-\u03baB\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-mlKGT6wBeik\/X29BpzZ0KFI\/AAAAAAAAfyE\/Uth0i3DrU7w9IFBGugeLk48MKKq3V_NPQCLcBGAsYHQ\/s204\/Clinical_Experimental_metastasis.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-mlKGT6wBeik\/X29BpzZ0KFI\/AAAAAAAAfyE\/Uth0i3DrU7w9IFBGugeLk48MKKq3V_NPQCLcBGAsYHQ\/s0\/Clinical_Experimental_metastasis.jpg\" border=\"0\" data-original-height=\"204\" data-original-width=\"153\" \/><\/a>Lee, G. R., Jang, S. H., Kim, C. J., Kim, A. R., Yoon, D. J., Park, N. H., &amp; Han, I. S. (2014).\u00a0<a href=\"https:\/\/link.springer.com\/article\/10.1007\/s10585-014-9678-x\">Capsaicin suppresses the migration of cholangiocarcinoma cells by down-regulating matrix metalloproteinase-9 expression via the AMPK\u2013NF-\u03baB signaling pathway<\/a>.\u00a0<i>Clinical &amp; experimental metastasis,<\/i>\u00a031(8), 897-907.<\/p>\n<p>El colangiocarcinoma es una de las neoplasias m\u00e1s dif\u00edciles de curar. Un factor pron\u00f3stico importante es la met\u00e1stasis, que excluye la resecci\u00f3n quir\u00fargica curativa. La evidencia reciente muestra que la capsaicina tiene un efecto inhibidor sobre la migraci\u00f3n e invasi\u00f3n de c\u00e9lulas cancerosas.<\/p>\n<p>Aqu\u00ed, investigamos el mecanismo molecular de los efectos anti-migraci\u00f3n y anti-invasi\u00f3n inducidos por capsaicina en las c\u00e9lulas del colangiocarcinoma HuCCT1.<\/p>\n<p>La migraci\u00f3n y la invasi\u00f3n se redujeron significativamente en respuesta a la capsaicina. La capsaicina tambi\u00e9n inhibi\u00f3 la expresi\u00f3n de la metaloproteinasa 9 de la matriz (MMP-9). En las c\u00e9lulas tratadas con capsaicina, aumentaron los niveles de AMPK fosforilada, y este efecto se elimin\u00f3 mediante el tratamiento con el inhibidor de AMPK, Compuesto C. La capsaicina aument\u00f3 la expresi\u00f3n de SIRT1, que puede activar el factor de transcripci\u00f3n NF-\u03baB mediante desacetilaci\u00f3n.<\/p>\n<p>Esto sugiere que la capsaicina activa el NF-\u03baB a trav\u00e9s de la v\u00eda SIRT1. Adem\u00e1s, la AMPK activada por capsaicina indujo la fosforilaci\u00f3n de I\u03baB\u03b1 y la localizaci\u00f3n nuclear de NF-\u03baB p65. Los ensayos de inmunoprecipitaci\u00f3n de cromatina demostraron que la capsaicina redujo la transcripci\u00f3n de MMP-9 inhibiendo la translocaci\u00f3n y desacetilaci\u00f3n de NF-\u03baB p65 a trav\u00e9s de SIRT1.<\/p>\n<p>Estos hallazgos proporcionan pruebas de que la capsaicina suprime la migraci\u00f3n y la invasi\u00f3n de las c\u00e9lulas del colangiocarcinoma al inhibir NF-\u03baB p65 a trav\u00e9s de las v\u00edas de se\u00f1alizaci\u00f3n AMPK-SIRT1 y AMPK-I\u03baB\u03b1, lo que conduce a la supresi\u00f3n posterior de la expresi\u00f3n de MMP-9.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Lee, G. R., Jang, S. H., Kim, C. J., Kim, A. R., Yoon, D. J., Park, N. H., &amp; Han, I. S. (2014).\u00a0Capsaicin suppresses the migration of cholangiocarcinoma cells by down-regulating matrix metalloproteinase-9 expression via the AMPK\u2013NF-\u03baB signaling pathway.\u00a0Clinical &amp; experimental metastasis,\u00a031(8), 897-907. El colangiocarcinoma es una de las neoplasias m\u00e1s dif\u00edciles de curar. Un [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-44092","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La capsaicina suprime la migraci\u00f3n de las c\u00e9lulas del colangiocarcinoma al regular negativamente la expresi\u00f3n de la metaloproteinasa-9 de la matriz a trav\u00e9s de la v\u00eda de se\u00f1alizaci\u00f3n AMPK-NF-\u03baB&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=44092\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La capsaicina suprime la migraci\u00f3n de las c\u00e9lulas del colangiocarcinoma al regular negativamente la expresi\u00f3n de la metaloproteinasa-9 de la matriz a trav\u00e9s de la v\u00eda de se\u00f1alizaci\u00f3n AMPK-NF-\u03baB&quot; -\" \/>\n<meta property=\"og:description\" content=\"Lee, G. R., Jang, S. H., Kim, C. J., Kim, A. R., Yoon, D. J., Park, N. H., &amp; Han, I. S. (2014).\u00a0Capsaicin suppresses the migration of cholangiocarcinoma cells by down-regulating matrix metalloproteinase-9 expression via the AMPK\u2013NF-\u03baB signaling pathway.\u00a0Clinical &amp; experimental metastasis,\u00a031(8), 897-907. El colangiocarcinoma es una de las neoplasias m\u00e1s dif\u00edciles de curar. 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