{"id":44114,"date":"2020-09-19T00:30:24","date_gmt":"2020-09-18T22:30:24","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=44114"},"modified":"2020-10-03T13:08:28","modified_gmt":"2020-10-03T11:08:28","slug":"44114","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=44114","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa activaci\u00f3n de AMPK inducida por berberina inhibe el potencial metast\u00e1sico de las c\u00e9lulas de melanoma mediante la reducci\u00f3n de la actividad de ERK y la expresi\u00f3n de la prote\u00edna COX-2\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-GKA5d98F5Fs\/X2-QknpFT3I\/AAAAAAAAfzY\/TYiIXMQF9LsC7EVCyNmzrRMPiDIT6LYJQCLcBGAsYHQ\/s259\/Biochemical_pharmacology.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-GKA5d98F5Fs\/X2-QknpFT3I\/AAAAAAAAfzY\/TYiIXMQF9LsC7EVCyNmzrRMPiDIT6LYJQCLcBGAsYHQ\/s0\/Biochemical_pharmacology.jpg\" border=\"0\" data-original-height=\"259\" data-original-width=\"194\" \/><\/a>Kim, H. S., Kim, M. J., Kim, E. J., Yang, Y., Lee, M. S., &amp; Lim, J. S. (2012). <a href=\"https:\/\/www.sciencedirect.com\/science\/article\/abs\/pii\/S0006295211008252\">Berberine-induced AMPK activation inhibits the metastatic potential of melanoma cells via reduction of ERK activity and COX-2 protein expression<\/a>.\u00a0<i>Biochemical pharmacology<\/i>, 83(3), 385-394.<\/p>\n<p>CONTEXTO: La berberina es un alcaloide de isoquinolina natural cl\u00ednicamente importante que afecta a diversas funciones biol\u00f3gicas, como la proliferaci\u00f3n, migraci\u00f3n y supervivencia celular. La activaci\u00f3n de la prote\u00edna quinasa activada por AMP (AMPK) regula la migraci\u00f3n de las c\u00e9lulas tumorales. Sin embargo, el papel espec\u00edfico de AMPK en el potencial metast\u00e1sico de las c\u00e9lulas cancerosas sigue siendo en gran parte desconocido.<\/p>\n<p>OBJETIVO DE LA INVESTIGACI\u00d3N: El presente estudio investig\u00f3 si la berberina induce la activaci\u00f3n de AMPK y si esta inducci\u00f3n afecta directamente a la migraci\u00f3n, adhesi\u00f3n e invasi\u00f3n de c\u00e9lulas de melanoma de rat\u00f3n.<\/p>\n<p>M\u00c9TODO \/ RESULTADOS: La berberina aument\u00f3 fuertemente la fosforilaci\u00f3n de AMPK a trav\u00e9s de la producci\u00f3n de especies reactivas de ox\u00edgeno (ROS). 5-aminoimidazol-4-carboxamida-1-\u03b2- d-ribofuran\u00f3sido (AICAR), un conocido activador de AMPK, tambi\u00e9n inhibi\u00f3 la adhesi\u00f3n e invasi\u00f3n de c\u00e9lulas tumorales y redujo la expresi\u00f3n de genes relacionados con la transici\u00f3n epitelial a mesenquimal (EMT). La eliminaci\u00f3n de las subunidades de AMPK\u03b1 mediante ARNip disminuy\u00f3 significativamente la inhibici\u00f3n de la invasi\u00f3n de c\u00e9lulas tumorales inducida por berberina. Adem\u00e1s, la berberina inhibi\u00f3 el potencial metast\u00e1sico de las c\u00e9lulas de melanoma a trav\u00e9s de una disminuci\u00f3n en la actividad de ERK y los niveles de prote\u00edna de la ciclooxigenasa-2 (COX-2) por una activaci\u00f3n de AMPK inducida por berberina. Estos datos se confirmaron utilizando un inhibidor espec\u00edfico de MEK, PD98059, y un inhibidor de COX-2, celecoxib. Los grupos tratados con berberina y AICAR demostraron una disminuci\u00f3n significativa de las met\u00e1stasis pulmonares en el modelo de met\u00e1stasis pulmonar in vivo. El tratamiento con berberina tambi\u00e9n redujo el potencial metast\u00e1sico de las c\u00e9lulas de melanoma humano A375.<\/p>\n<p>CONCLUSI\u00d3N: En conjunto, nuestros resultados sugieren que la activaci\u00f3n de AMPK inducida por berberina inhibe el potencial metast\u00e1sico de las c\u00e9lulas tumorales a trav\u00e9s de una reducci\u00f3n en la actividad de la v\u00eda de se\u00f1alizaci\u00f3n ERK y los niveles de prote\u00edna COX-2.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Kim, H. S., Kim, M. J., Kim, E. J., Yang, Y., Lee, M. S., &amp; Lim, J. S. (2012). Berberine-induced AMPK activation inhibits the metastatic potential of melanoma cells via reduction of ERK activity and COX-2 protein expression.\u00a0Biochemical pharmacology, 83(3), 385-394. CONTEXTO: La berberina es un alcaloide de isoquinolina natural cl\u00ednicamente importante que afecta a [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-44114","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La activaci\u00f3n de AMPK inducida por berberina inhibe el potencial metast\u00e1sico de las c\u00e9lulas de melanoma mediante la reducci\u00f3n de la actividad de ERK y la expresi\u00f3n de la prote\u00edna COX-2&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=44114\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La activaci\u00f3n de AMPK inducida por berberina inhibe el potencial metast\u00e1sico de las c\u00e9lulas de melanoma mediante la reducci\u00f3n de la actividad de ERK y la expresi\u00f3n de la prote\u00edna COX-2&quot; -\" \/>\n<meta property=\"og:description\" content=\"Kim, H. S., Kim, M. J., Kim, E. J., Yang, Y., Lee, M. S., &amp; Lim, J. S. (2012). Berberine-induced AMPK activation inhibits the metastatic potential of melanoma cells via reduction of ERK activity and COX-2 protein expression.\u00a0Biochemical pharmacology, 83(3), 385-394. 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inhibe el potencial metast\u00e1sico de las c\u00e9lulas de melanoma mediante la reducci\u00f3n de la actividad de ERK y la expresi\u00f3n de la prote\u00edna COX-2\" -","robots":{"index":"index","follow":"follow","max-snippet":"max-snippet:-1","max-image-preview":"max-image-preview:large","max-video-preview":"max-video-preview:-1"},"canonical":"https:\/\/rina.naturopatiadigital.eu\/?p=44114","og_locale":"es_ES","og_type":"article","og_title":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \"La activaci\u00f3n de AMPK inducida por berberina inhibe el potencial metast\u00e1sico de las c\u00e9lulas de melanoma mediante la reducci\u00f3n de la actividad de ERK y la expresi\u00f3n de la prote\u00edna COX-2\" -","og_description":"Kim, H. S., Kim, M. J., Kim, E. J., Yang, Y., Lee, M. S., &amp; Lim, J. S. (2012). Berberine-induced AMPK activation inhibits the metastatic potential of melanoma cells via reduction of ERK activity and COX-2 protein expression.\u00a0Biochemical pharmacology, 83(3), 385-394. CONTEXTO: La berberina es un alcaloide de isoquinolina natural cl\u00ednicamente importante que afecta a [&hellip;]","og_url":"https:\/\/rina.naturopatiadigital.eu\/?p=44114","article_published_time":"2020-09-18T22:30:24+00:00","article_modified_time":"2020-10-03T11:08:28+00:00","og_image":[{"url":"https:\/\/1.bp.blogspot.com\/-GKA5d98F5Fs\/X2-QknpFT3I\/AAAAAAAAfzY\/TYiIXMQF9LsC7EVCyNmzrRMPiDIT6LYJQCLcBGAsYHQ\/s0\/Biochemical_pharmacology.jpg"}],"author":"admin","twitter_card":"summary_large_image","twitter_misc":{"Escrito por":"admin","Tiempo de lectura":"2 minutos"},"schema":{"@context":"https:\/\/schema.org","@graph":[{"@type":"Article","@id":"https:\/\/rina.naturopatiadigital.eu\/?p=44114#article","isPartOf":{"@id":"https:\/\/rina.naturopatiadigital.eu\/?p=44114"},"author":{"name":"admin","@id":"https:\/\/rina.naturopatiadigital.eu\/#\/schema\/person\/432852c9ed996fc42e869a813ecbffd7"},"headline":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: 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