{"id":44401,"date":"2020-10-12T04:30:50","date_gmt":"2020-10-12T02:30:50","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=44401"},"modified":"2020-10-13T19:36:56","modified_gmt":"2020-10-13T17:36:56","slug":"area-de-conocimiento-tecnologia-naturopatica-o-naturopatia-aplicada-modulo-naturopatia-fitocomplementaria-herbologia-el-polifenol-epigalocatequina-3-galato-del-te-verde-bloquea-la-activa","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=44401","title":{"rendered":"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria &#8211; HERBOLOGIA: \u00abEl polifenol (-) &#8211; epigalocatequina-3-galato del t\u00e9 verde bloquea la activaci\u00f3n del factor nuclear kappa B al inhibir la actividad de la quinasa I kappa B en la l\u00ednea de c\u00e9lulas epiteliales intestinales IEC-6\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-RIOKcvXrmzo\/X4XkY1V9hlI\/AAAAAAAAgFM\/0Mo_8GQH0iMBYQ5IhENOs1kQTP1GtPYfwCLcBGAsYHQ\/s220\/Molecular_Pharmacology.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-RIOKcvXrmzo\/X4XkY1V9hlI\/AAAAAAAAgFM\/0Mo_8GQH0iMBYQ5IhENOs1kQTP1GtPYfwCLcBGAsYHQ\/s0\/Molecular_Pharmacology.jpg\" border=\"0\" data-original-height=\"220\" data-original-width=\"164\" \/><\/a>Yang, F., Oz, H. S., Barve, S., De Villiers, W. J., McClain, C. J., &amp; Varilek, G. W. (2001).\u00a0<a href=\"https:\/\/scholar.google.com\/scholar_url?url=https:\/\/www.researchgate.net\/profile\/Helieh_Oz\/publication\/11841846_The_Green_Tea_Polyphenol_--Epigallocatechin-3-Gallate_Blocks_Nuclear_Factor-kB_Activation_by_Inhibiting_IkB_Kinase_Activity_in_the_Intestinal_Epithelial_Cell_Line_IEC-6\/links\/5a41bcf50f7e9ba868a19d2d\/The-Green-Tea-Polyphenol--Epigallocatechin-3-Gallate-Blocks-Nuclear-Factor-kB-Activation-by-Inhibiting-IkB-Kinase-Activity-in-the-Intestinal-Epithelial-Cell-Line-IEC-6.pdf&amp;hl=es&amp;sa=T&amp;oi=gsb-gga&amp;ct=res&amp;cd=0&amp;d=3552769524524835086&amp;ei=C-WFX9SlG--Qy9YPmPqiqAY&amp;scisig=AAGBfm3qFniywY5P054Op9s-85xdZVEh1g\">The green tea polyphenol (\u2212)-epigallocatechin-3-gallate blocks nuclear factor-\u03baB activation by inhibiting I\u03baB kinase activity in the intestinal epithelial cell line IEC-6<\/a>.\u00a0<i>Molecular Pharmacology<\/i>, 60(3), 528-533.<\/p>\n<p>El complejo de quinasa I kappa B (IKK) media la activaci\u00f3n del factor de transcripci\u00f3n factor nuclear kappa B (NF-kappa B). Anteriormente mostramos que los polifenoles del t\u00e9 verde inhib\u00edan la producci\u00f3n del factor de necrosis tumoral alfa (TNF alfa) mediada por endotoxinas al bloquear la activaci\u00f3n de NF-kappa B.<\/p>\n<p>En este estudio, evaluamos si los polifenoles del t\u00e9 verde inhiben NF-kappa B al bloquear la actividad de IKK.<\/p>\n<p>Evaluamos la actividad de IKK mediante la detecci\u00f3n de cambios en la fosforilaci\u00f3n de una prote\u00edna de fusi\u00f3n I kappa B alfa-glutati\u00f3n S-transferasa (GST). Las c\u00e9lulas IEC-6 pretratadas con un extracto de polifenoles de t\u00e9 verde (GrTP; 0-0,4 mg \/ ml) ten\u00edan una actividad disminuida de IKK y NF-kappa B inducida por TNF alfa.<\/p>\n<p>De los diversos GrTP, (-) &#8211; epigalocatequina-3-galato (EGCG) fue el inhibidor m\u00e1s potente. A continuaci\u00f3n, examinamos si EGCG inhib\u00eda la IKK activada. En extractos citos\u00f3licos de c\u00e9lulas estimuladas con TNF alfa, EGCG inhibi\u00f3 la fosforilaci\u00f3n de I kappa B alfa-GST (IC (50)&gt; 18 microM) consistente con la inhibici\u00f3n de la actividad IKK.<\/p>\n<p>Usando otros polifenoles, demostramos que el grupo galato era esencial para la inhibici\u00f3n y que los antioxidantes no eran efectivos para bloquear la IKK activada. Es importante destacar que EGCG disminuy\u00f3 la actividad de IKK en extractos citos\u00f3licos de c\u00e9lulas transfectadas con NIK de forma transitoria. Este \u00faltimo hallazgo mostr\u00f3 que nuestros hallazgos no estaban relacionados con la actividad quinasa inespec\u00edfica.<\/p>\n<p>En conclusi\u00f3n, EGCG es un inhibidor eficaz de la actividad de IKK. Esto puede explicar, al menos en parte, algunos de los efectos antiinflamatorios y anticancerosos del t\u00e9 verde.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Yang, F., Oz, H. S., Barve, S., De Villiers, W. J., McClain, C. J., &amp; Varilek, G. W. (2001).\u00a0The green tea polyphenol (\u2212)-epigallocatechin-3-gallate blocks nuclear factor-\u03baB activation by inhibiting I\u03baB kinase activity in the intestinal epithelial cell line IEC-6.\u00a0Molecular Pharmacology, 60(3), 528-533. El complejo de quinasa I kappa B (IKK) media la activaci\u00f3n del factor [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[5],"tags":[],"class_list":["post-44401","post","type-post","status-publish","format-standard","hentry","category-naturopatia-fitocomplementaria-herbologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;El polifenol (-) - epigalocatequina-3-galato del t\u00e9 verde bloquea la activaci\u00f3n del factor nuclear kappa B al inhibir la actividad de la quinasa I kappa B en la l\u00ednea de c\u00e9lulas epiteliales intestinales IEC-6&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=44401\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;El polifenol (-) - epigalocatequina-3-galato del t\u00e9 verde bloquea la activaci\u00f3n del factor nuclear kappa B al inhibir la actividad de la quinasa I kappa B en la l\u00ednea de c\u00e9lulas epiteliales intestinales IEC-6&quot; -\" \/>\n<meta property=\"og:description\" content=\"Yang, F., Oz, H. S., Barve, S., De Villiers, W. J., McClain, C. J., &amp; Varilek, G. W. (2001).\u00a0The green tea polyphenol (\u2212)-epigallocatechin-3-gallate blocks nuclear factor-\u03baB activation by inhibiting I\u03baB kinase activity in the intestinal epithelial cell line IEC-6.\u00a0Molecular Pharmacology, 60(3), 528-533. 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S., Barve, S., De Villiers, W. J., McClain, C. J., &amp; Varilek, G. W. (2001).\u00a0The green tea polyphenol (\u2212)-epigallocatechin-3-gallate blocks nuclear factor-\u03baB activation by inhibiting I\u03baB kinase activity in the intestinal epithelial cell line IEC-6.\u00a0Molecular Pharmacology, 60(3), 528-533. 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