{"id":44445,"date":"2020-10-17T05:30:19","date_gmt":"2020-10-17T03:30:19","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=44445"},"modified":"2020-10-18T23:12:46","modified_gmt":"2020-10-18T21:12:46","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-el-acido-ursolico-previene-el-aumento-de-la-inflamacion-periferica-y-la-hiperalgesia-inflamatoria-en-ratas-obesas-inducidas-por","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=44445","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abEl \u00e1cido urs\u00f3lico previene el aumento de la inflamaci\u00f3n perif\u00e9rica y la hiperalgesia inflamatoria en ratas obesas inducidas por una dieta alta en grasas al restaurar PPAR\u03b1 espinal regulado negativamente\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-f_dOLobSwK4\/X4yvG45v03I\/AAAAAAAAgQY\/YvsqzonZ2_4V904aPgf7bGnYWdyvQfArACLcBGAsYHQ\/s209\/Molecular_Medicine%2BReports.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-f_dOLobSwK4\/X4yvG45v03I\/AAAAAAAAgQY\/YvsqzonZ2_4V904aPgf7bGnYWdyvQfArACLcBGAsYHQ\/s0\/Molecular_Medicine%2BReports.jpg\" border=\"0\" data-original-height=\"209\" data-original-width=\"151\" \/><\/a>Zhang, Y., Song, C., Li, H., Hou, J., &amp; Li, D. (2016). <a href=\"https:\/\/www.spandidos-publications.com\/mmr\/13\/6\/5309?text=fulltext\">Ursolic acid prevents augmented peripheral inflammation and inflammatory hyperalgesia in high-fat diet-induced obese rats by restoring downregulated spinal PPAR\u03b1<\/a>.<i>\u00a0Molecular Medicine Reports<\/i>, 13(6), 5309-5316.<\/p>\n<p>La obesidad es un factor de riesgo para varios s\u00edndromes de dolor y est\u00e1 asociada con una mayor sensibilidad al dolor. La evidencia sugiere que la obesidad causa la regulaci\u00f3n a la baja del receptor activado por proliferador de peroxisoma (PPAR) \u03b1 en la m\u00e9dula espinal, lo que contribuye al aumento del edema perif\u00e9rico y la hiperalgesia inflamatoria. Se ha demostrado que el \u00e1cido urs\u00f3lico (UA), un \u00e1cido carbox\u00edlico triterpenoide pentac\u00edclico natural, regula positivamente el PPAR\u03b1 en los tejidos perif\u00e9ricos de los animales obesos.<\/p>\n<p>El presente estudio plante\u00f3 la hip\u00f3tesis de que la AU previene el aumento de la inflamaci\u00f3n perif\u00e9rica y la hiperalgesia inflamatoria en la obesidad al restaurar PPAR\u03b1 espinal regulado negativamente.<\/p>\n<p>El presente estudio demostr\u00f3 que las ratas Sprague-Dawley alimentadas con una dieta alta en grasas (HFD) durante 12 semanas desarrollaron obesidad y trastornos metab\u00f3licos. Despu\u00e9s de la inyecci\u00f3n de carragenina, las ratas HFD mostraron un aumento de la hiperalgesia t\u00e9rmica y el edema de las patas. en comparaci\u00f3n con las ratas alimentadas con una dieta baja en grasas.<\/p>\n<p>Las investigaciones moleculares revelaron que las ratas HFD mostraron una disminuci\u00f3n de la actividad de PPAR\u03b1 y una expresi\u00f3n exagerada de mediadores inflamatorios y actividad del factor nuclear-kB en la m\u00e9dula espinal en respuesta al carragenano. La administraci\u00f3n oral de UA mejor\u00f3 la obesidad y el trastorno metab\u00f3lico y previno el aumento de la hiperalgesia t\u00e9rmica y el edema de las patas en las ratas HFD. Adem\u00e1s, UA normaliz\u00f3 la actividad de PPAR\u03b1 e inhibi\u00f3 la respuesta inflamatoria exagerada de la m\u00e9dula espinal al carragenano. Aunque la eliminaci\u00f3n de PPAR\u03b1 espinal con ARN de interferencia peque\u00f1o despu\u00e9s de la administraci\u00f3n de UA no alter\u00f3 la obesidad o los par\u00e1metros metab\u00f3licos, erradic\u00f3 los efectos beneficiosos de UA sobre la hiperalgesia t\u00e9rmica y el edema de la pata, y revirti\u00f3 la respuesta inflamatoria de la m\u00e9dula espinal.<\/p>\n<p>Estos resultados sugirieron que la administraci\u00f3n sist\u00e9mica de UA inhibi\u00f3 la respuesta inflamatoria exagerada de la m\u00e9dula espinal a la estimulaci\u00f3n inflamatoria perif\u00e9rica en la obesidad inducida por HFD al restaurar PPAR\u03b1 espinal regulado a la baja, previniendo la inflamaci\u00f3n perif\u00e9rica y la hiperalgesia inflamatoria. La AU puede ser una opci\u00f3n terap\u00e9utica potencial para la prevenci\u00f3n del aumento del dolor inflamatorio en pacientes obesos.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Zhang, Y., Song, C., Li, H., Hou, J., &amp; Li, D. (2016). Ursolic acid prevents augmented peripheral inflammation and inflammatory hyperalgesia in high-fat diet-induced obese rats by restoring downregulated spinal PPAR\u03b1.\u00a0Molecular Medicine Reports, 13(6), 5309-5316. La obesidad es un factor de riesgo para varios s\u00edndromes de dolor y est\u00e1 asociada con una mayor sensibilidad al [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-44445","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El \u00e1cido urs\u00f3lico previene el aumento de la inflamaci\u00f3n perif\u00e9rica y la hiperalgesia inflamatoria en ratas obesas inducidas por una dieta alta en grasas al restaurar PPAR\u03b1 espinal regulado negativamente&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=44445\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El \u00e1cido urs\u00f3lico previene el aumento de la inflamaci\u00f3n perif\u00e9rica y la hiperalgesia inflamatoria en ratas obesas inducidas por una dieta alta en grasas al restaurar PPAR\u03b1 espinal regulado negativamente&quot; -\" \/>\n<meta property=\"og:description\" content=\"Zhang, Y., Song, C., Li, H., Hou, J., &amp; Li, D. 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