{"id":45098,"date":"2020-12-07T01:30:15","date_gmt":"2020-12-07T00:30:15","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=45098"},"modified":"2020-12-06T12:32:40","modified_gmt":"2020-12-06T11:32:40","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-la-tomatidina-reprime-la-invasion-y-migracion-de-las-celulas-u2os-y-hos-del-osteosarcoma-humano-mediante-la-supresion-de-la-pre","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=45098","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa tomatidina reprime la invasi\u00f3n y migraci\u00f3n de las c\u00e9lulas U2OS y HOS del osteosarcoma humano mediante la supresi\u00f3n de la presenilina 1 y la v\u00eda c-Raf-MEK-ERK\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-Tnnv_49e_Bc\/X8zAcPjyDaI\/AAAAAAAAhDw\/slo_Pi70XegNjDRxBI1dnGzWwyWrlyw9ACLcBGAsYHQ\/s855\/Molecules2.png\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-Tnnv_49e_Bc\/X8zAcPjyDaI\/AAAAAAAAhDw\/slo_Pi70XegNjDRxBI1dnGzWwyWrlyw9ACLcBGAsYHQ\/s320\/Molecules2.png\" height=\"320\" border=\"0\" data-original-height=\"855\" data-original-width=\"596\" \/><\/a>Hsieh, M. H., Yang, J. S., Lin, R. C., Hsieh, Y. H., Yang, S. F., Chang, H. R., &amp; Lu, K. H. (2020). <a href=\"https:\/\/www.mdpi.com\/1420-3049\/25\/2\/326\/htm\">Tomatidine Represses Invasion and Migration of Human Osteosarcoma U2OS and HOS Cells by Suppression of Presenilin 1 and c-Raf\u2013MEK\u2013ERK Pathway<\/a><i>. Molecules<\/i>, 25(2), 326.<\/p>\n<p>CONTEXTO: El osteosarcoma, que es el tumor \u00f3seo maligno m\u00e1s prevalente, es responsable de la gran mayor\u00eda de las muertes asociadas al c\u00e1ncer de hueso debido a su alto potencial metast\u00e1sico. Aunque se sugiere que la tomatidina sirve como quimiosensibilizador en tumores resistentes a m\u00faltiples f\u00e1rmacos, a\u00fan se desconoce el efecto antimetast\u00e1sico de la tomatidina en el osteosarcoma.<\/p>\n<p>OBJETIVO: Aqu\u00ed, probamos la hip\u00f3tesis de que la tomatidina suprime la migraci\u00f3n y la invasi\u00f3n, caracter\u00edsticas que est\u00e1n asociadas con el proceso metast\u00e1sico en las c\u00e9lulas de osteosarcoma humano y tambi\u00e9n investigamos su v\u00eda subyacente.<\/p>\n<p>METODO \/ RESULTADOS: La tomatidina, hasta 100 \u03bcM, sin citotoxicidad, inhibi\u00f3 la capacidad de invasi\u00f3n y migraci\u00f3n de las c\u00e9lulas U2OS y HOS del osteosarcoma humano y reprimi\u00f3 la expresi\u00f3n de presenilina 1 (PS-1) de las c\u00e9lulas U2OS. Despu\u00e9s de la ca\u00edda de PS-1, los comportamientos biol\u00f3gicos de invasi\u00f3n celular y potencial migratorio de las c\u00e9lulas U2OS y HOS se redujeron significativamente. Si bien la tomatidina disminuy\u00f3 significativamente la fosforilaci\u00f3n de c-Raf, quinasa regulada por se\u00f1al mit\u00f3gena \/ extracelular (MEK) y prote\u00edna quinasa regulada por se\u00f1al extracelular (ERK) 1\/2 en las c\u00e9lulas U2OS, no hay influencias obvias sobre la quinasa p-Jun N-terminal , p38 y Akt, incluida su fosforilaci\u00f3n, se observaron. En ERK 1 que silencia las c\u00e9lulas U2 OS, la tomatidina mejor\u00f3 a\u00fan m\u00e1s la disminuci\u00f3n de su potencial migratorio y actividades invasivas.<\/p>\n<p>CONCLUSION: Concluimos que tanto el PS-1 derivado de las c\u00e9lulas U2OS y HOS como la v\u00eda c-Raf-MEK-ERK contribuyen a la invasi\u00f3n y migraci\u00f3n celular y la tomatidina podr\u00eda inhibir los fen\u00f3menos. Estos hallazgos indican que la tomatidina podr\u00eda ser un candidato potencial para el tratamiento anti-met\u00e1stasis del osteosarcoma humano.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Hsieh, M. H., Yang, J. S., Lin, R. C., Hsieh, Y. H., Yang, S. F., Chang, H. R., &amp; Lu, K. H. (2020). Tomatidine Represses Invasion and Migration of Human Osteosarcoma U2OS and HOS Cells by Suppression of Presenilin 1 and c-Raf\u2013MEK\u2013ERK Pathway. Molecules, 25(2), 326. CONTEXTO: El osteosarcoma, que es el tumor \u00f3seo maligno [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-45098","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La tomatidina reprime la invasi\u00f3n y migraci\u00f3n de las c\u00e9lulas U2OS y HOS del osteosarcoma humano mediante la supresi\u00f3n de la presenilina 1 y la v\u00eda c-Raf-MEK-ERK&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=45098\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;La tomatidina reprime la invasi\u00f3n y migraci\u00f3n de las c\u00e9lulas U2OS y HOS del osteosarcoma humano mediante la supresi\u00f3n de la presenilina 1 y la v\u00eda c-Raf-MEK-ERK&quot; -\" \/>\n<meta property=\"og:description\" content=\"Hsieh, M. H., Yang, J. S., Lin, R. C., Hsieh, Y. H., Yang, S. F., Chang, H. R., &amp; Lu, K. H. (2020). Tomatidine Represses Invasion and Migration of Human Osteosarcoma U2OS and HOS Cells by Suppression of Presenilin 1 and c-Raf\u2013MEK\u2013ERK Pathway. Molecules, 25(2), 326. CONTEXTO: El osteosarcoma, que es el tumor \u00f3seo maligno [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=45098\" \/>\n<meta property=\"article:published_time\" content=\"2020-12-07T00:30:15+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2020-12-06T11:32:40+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-Tnnv_49e_Bc\/X8zAcPjyDaI\/AAAAAAAAhDw\/slo_Pi70XegNjDRxBI1dnGzWwyWrlyw9ACLcBGAsYHQ\/s320\/Molecules2.png\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" content=\"Tiempo de lectura\" \/>\n\t<meta name=\"twitter:data2\" content=\"2 minutos\" \/>\n<script type=\"application\/ld+json\" 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H., Yang, J. S., Lin, R. C., Hsieh, Y. H., Yang, S. F., Chang, H. R., &amp; Lu, K. H. (2020). Tomatidine Represses Invasion and Migration of Human Osteosarcoma U2OS and HOS Cells by Suppression of Presenilin 1 and c-Raf\u2013MEK\u2013ERK Pathway. Molecules, 25(2), 326. CONTEXTO: El osteosarcoma, que es el tumor \u00f3seo maligno [&hellip;]","og_url":"https:\/\/rina.naturopatiadigital.eu\/?p=45098","article_published_time":"2020-12-07T00:30:15+00:00","article_modified_time":"2020-12-06T11:32:40+00:00","og_image":[{"url":"https:\/\/1.bp.blogspot.com\/-Tnnv_49e_Bc\/X8zAcPjyDaI\/AAAAAAAAhDw\/slo_Pi70XegNjDRxBI1dnGzWwyWrlyw9ACLcBGAsYHQ\/s320\/Molecules2.png"}],"author":"admin","twitter_card":"summary_large_image","twitter_misc":{"Escrito por":"admin","Tiempo de lectura":"2 minutos"},"schema":{"@context":"https:\/\/schema.org","@graph":[{"@type":"Article","@id":"https:\/\/rina.naturopatiadigital.eu\/?p=45098#article","isPartOf":{"@id":"https:\/\/rina.naturopatiadigital.eu\/?p=45098"},"author":{"name":"admin","@id":"https:\/\/rina.naturopatiadigital.eu\/#\/schema\/person\/432852c9ed996fc42e869a813ecbffd7"},"headline":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abLa tomatidina reprime la invasi\u00f3n y 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