{"id":45259,"date":"2020-12-21T06:30:31","date_gmt":"2020-12-21T05:30:31","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=45259"},"modified":"2020-12-23T13:21:42","modified_gmt":"2020-12-23T12:21:42","slug":"area-de-conocimiento-tecnologia-naturopatica-o-naturopatia-aplicada-modulo-naturopatia-fitocomplementaria-herbologia-la-apigenina-un-componente-de-las-flores-de-matricaria-recutita-es-un-lig","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=45259","title":{"rendered":"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria &#8211; HERBOLOGIA: \u00abLa apigenina, un componente de las flores de Matricaria recutita, es un ligando central de receptores de benzodiazepinas con efectos ansiol\u00edticos\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-WrPc51915Vo\/X-M1tLcV4OI\/AAAAAAAAhUY\/sViKTRvn-4UleGiYRwFNunelkZb2Yx9FgCLcBGAsYHQ\/s256\/Planta_Medica.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-WrPc51915Vo\/X-M1tLcV4OI\/AAAAAAAAhUY\/sViKTRvn-4UleGiYRwFNunelkZb2Yx9FgCLcBGAsYHQ\/s0\/Planta_Medica.jpg\" border=\"0\" data-original-height=\"256\" data-original-width=\"197\" \/><\/a>Viola, H., Wasowski, C., De Stein, M. L., Wolfman, C., Silveira, R., Dajas, F., &#8230; &amp; Paladini, A. C. (1995). <a href=\"https:\/\/www.thieme-connect.com\/products\/ejournals\/abstract\/10.1055\/s-2006-958058\">Apigenin, a component of Matricaria recutita flowers, is a central benzodiazepine receptors-ligand with anxiolytic effects<\/a>.<i>\u00a0Planta medica<\/i>, 61(03), 213-216.<\/p>\n<p>Las cabezas de flores secas de Matricaria recutita L. (Asteraceae) se utilizan en la medicina popular para preparar un t\u00e9 espasmol\u00edtico y sedante.<\/p>\n<p>Nuestro fraccionamiento del extracto acuoso de esta planta permiti\u00f3 la detecci\u00f3n de varias fracciones con importante afinidad por el receptor central de benzodiazepinas y el aislamiento e identificaci\u00f3n de 5,7,4\u2032-trihidroxiflavona (apigenina) en una de ellas.<\/p>\n<p>La apigenina inhibi\u00f3 competitivamente la uni\u00f3n de flunitrazepam con una Ki de 4 \u00b5M y no tuvo ning\u00fan efecto sobre los receptores muscar\u00ednicos, los receptores adren\u00e9rgicos \u03b11 y sobre la uni\u00f3n del muscimol a los receptores GABAA.<\/p>\n<p>La apigenina tuvo una clara actividad ansiol\u00edtica en ratones en el laberinto positivo elevado sin evidenciar sedaci\u00f3n o efectos relajantes musculares a dosis similares a las utilizadas para las benzodiazepinas cl\u00e1sicas y no se detect\u00f3 acci\u00f3n anticonvulsiva. Sin embargo, un aumento de 10 veces en la dosis produjo un leve efecto sedante ya que fue evidente una reducci\u00f3n del 26% en la actividad locomotora ambulatoria y una disminuci\u00f3n del 35% en los par\u00e1metros de la tabla de agujeros.<\/p>\n<p>Los resultados reportados en este trabajo demuestran que la apigenina es un ligando de los receptores centrales de benzodiazepina que ejerce efectos ansiol\u00edticos y sedantes leves, pero no es anticonvulsivante ni miorrelajante.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Viola, H., Wasowski, C., De Stein, M. L., Wolfman, C., Silveira, R., Dajas, F., &#8230; &amp; Paladini, A. C. (1995). Apigenin, a component of Matricaria recutita flowers, is a central benzodiazepine receptors-ligand with anxiolytic effects.\u00a0Planta medica, 61(03), 213-216. Las cabezas de flores secas de Matricaria recutita L. (Asteraceae) se utilizan en la medicina popular para [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[5],"tags":[],"class_list":["post-45259","post","type-post","status-publish","format-standard","hentry","category-naturopatia-fitocomplementaria-herbologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;La apigenina, un componente de las flores de Matricaria recutita, es un ligando central de receptores de benzodiazepinas con efectos ansiol\u00edticos&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=45259\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;La apigenina, un componente de las flores de Matricaria recutita, es un ligando central de receptores de benzodiazepinas con efectos ansiol\u00edticos&quot; -\" \/>\n<meta property=\"og:description\" content=\"Viola, H., Wasowski, C., De Stein, M. L., Wolfman, C., Silveira, R., Dajas, F., &#8230; &amp; Paladini, A. C. (1995). Apigenin, a component of Matricaria recutita flowers, is a central benzodiazepine receptors-ligand with anxiolytic effects.\u00a0Planta medica, 61(03), 213-216. Las cabezas de flores secas de Matricaria recutita L. 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