{"id":45273,"date":"2020-12-22T06:30:13","date_gmt":"2020-12-22T05:30:13","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=45273"},"modified":"2020-12-24T22:12:05","modified_gmt":"2020-12-24T21:12:05","slug":"area-de-conocimiento-tecnologia-naturopatica-o-naturopatia-aplicada-modulo-naturopatia-fitocomplementaria-herbologia-black-cohosh-actua-como-ligando-competitivo-mixto-y-agonista-parcial-del-re","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=45273","title":{"rendered":"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria &#8211; HERBOLOGIA: \u00abBlack Cohosh act\u00faa como ligando competitivo mixto y agonista parcial del receptor de serotonina\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-sv2JsWsRb9Y\/X-UDSzGna0I\/AAAAAAAAhV8\/hiPDFrNq1wUU8Q51PdWxlk3e6CY51UW7gCLcBGAsYHQ\/s397\/Journal_Agricultural%2Band%2BFood%2BChemistry.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-sv2JsWsRb9Y\/X-UDSzGna0I\/AAAAAAAAhV8\/hiPDFrNq1wUU8Q51PdWxlk3e6CY51UW7gCLcBGAsYHQ\/s320\/Journal_Agricultural%2Band%2BFood%2BChemistry.jpg\" height=\"320\" border=\"0\" data-original-height=\"397\" data-original-width=\"299\" \/><\/a>Burdette, J. E., Liu, J., Chen, S. N., Fabricant, D. S., Piersen, C. E., Barker, E. L., &#8230; &amp; Bolton, J. L. (2003). <a href=\"https:\/\/pubs.acs.org\/doi\/abs\/10.1021\/jf034264r\">Black cohosh acts as a mixed competitive ligand and partial agonist of the serotonin receptor<\/a>.\u00a0<i>Journal of Agricultural and Food Chemistry<\/i>, 51(19), 5661-5670.<\/p>\n<p>OBJETIVO: Extractos del rizoma de cohosh negro [ Actaea racemosa L., antes llamado Cimicifuga racemosa(L.) Nutt.] fueron evaluados por posibles mecanismos de acci\u00f3n en el alivio de los sofocos menop\u00e1usicos.<\/p>\n<p>METODOLOGIA: Se administr\u00f3 a ratas Sprague-Dawley ovariectomizadas un extracto de cohosh negro de 2-propanol al 40% [4, 40 y 400 mg \/ (kg \u00b7 d\u00eda)] por sonda durante 2 semanas con o sin estradiol [50 \u03bcg \/ (kg \u00b7 d\u00eda) ] para determinar si el cohosh negro podr\u00eda actuar como estr\u00f3geno o antiestr\u00f3geno sobre la base de un aumento en el peso uterino o cornificaci\u00f3n celular vaginal. No se observaron efectos sobre el peso uterino o sobre la cornificaci\u00f3n celular vaginal en ratas tratadas con cohosh negro solo o en combinaci\u00f3n con 17\u03b2-estradiol, lo que indica que este extracto de cohosh negro no ten\u00eda propiedades estrog\u00e9nicas o antiestrog\u00e9nicas en el modelo de rata ovariectomizada. Para evaluar otras posibles v\u00edas por las cuales el cohosh negro podr\u00eda reducir los sofocos menop\u00e1usicos, la actividad de la serotonina se evalu\u00f3 primero mediante la inhibici\u00f3n de la uni\u00f3n del radioligando a preparaciones de membranas celulares que contienen subtipos de receptores de serotonina humana recombinantes (5-HT). Se prob\u00f3 un extracto de cohosh negro de 2-propanol al 40% contra 10 subtipos del receptor de serotonina, revelando la presencia de compuestos con fuerte uni\u00f3n al 5-HT.Subtipos 1A , 5-HT 1D y 5-HT 7 . Los estudios de uni\u00f3n posteriores se llevaron a cabo utilizando receptores 5-HT 1A y 5-HT 7 debido a su asociaci\u00f3n con el hipot\u00e1lamo, que se ha implicado en la generaci\u00f3n de sofocos.<\/p>\n<p>RESULTADOS: El extracto de cohosh negro al 40% 2-propanol inhibi\u00f3 la uni\u00f3n de la dietilamida del \u00e1cido lis\u00e9rgico [ 3 H] (LSD) al receptor humano 5-HT 7 (IC 50 = 2,4 \u00b1 0,4 \u03bcg \/ ml) con mayor potencia que la uni\u00f3n de [ 3 H] -8-hidroxi-2- (di- N -propilamino) tetralina al receptor 5-HT 1A de rata (IC 50= 13,9 \u00b1 0,6 \u03bcg \/ ml). An\u00e1lisis de los datos de uni\u00f3n a ligando indica que los componentes de un extracto de metanol cohosh negro funcionaban como un ligando competitivo mixto de la 5-HT 7 receptor. Adem\u00e1s, un extracto de metanol cohosh negro eleva los niveles de AMPc en 293T-5-HT 7 c\u00e9lulas HEK transfectadas, lo que sugiere el extracto actuado como un agonista parcial en el receptor. La elevaci\u00f3n de cAMP mediada por el extracto de cohosh negro podr\u00eda revertirse en presencia del antagonista metiotepina, lo que indica un proceso mediado por receptores.<\/p>\n<p>CONCLUSION: Estos datos sugieren que las reducciones en los sofocos en algunas mujeres que toman cohosh negro pueden no deberse a propiedades estrog\u00e9nicas. Este estudio identifica otros posibles objetivos biol\u00f3gicos del cohosh negro que podr\u00edan explicar los efectos biol\u00f3gicos informados.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Burdette, J. E., Liu, J., Chen, S. N., Fabricant, D. S., Piersen, C. E., Barker, E. L., &#8230; &amp; Bolton, J. L. (2003). Black cohosh acts as a mixed competitive ligand and partial agonist of the serotonin receptor.\u00a0Journal of Agricultural and Food Chemistry, 51(19), 5661-5670. OBJETIVO: Extractos del rizoma de cohosh negro [ Actaea racemosa [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[5],"tags":[],"class_list":["post-45273","post","type-post","status-publish","format-standard","hentry","category-naturopatia-fitocomplementaria-herbologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;Black Cohosh act\u00faa como ligando competitivo mixto y agonista parcial del receptor de serotonina&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=45273\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;Black Cohosh act\u00faa como ligando competitivo mixto y agonista parcial del receptor de serotonina&quot; -\" \/>\n<meta property=\"og:description\" content=\"Burdette, J. E., Liu, J., Chen, S. N., Fabricant, D. S., Piersen, C. E., Barker, E. L., &#8230; &amp; Bolton, J. L. (2003). Black cohosh acts as a mixed competitive ligand and partial agonist of the serotonin receptor.\u00a0Journal of Agricultural and Food Chemistry, 51(19), 5661-5670. 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