{"id":45278,"date":"2020-12-23T01:30:18","date_gmt":"2020-12-23T00:30:18","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=45278"},"modified":"2020-12-25T10:39:57","modified_gmt":"2020-12-25T09:39:57","slug":"cohosh-negro-actaea-racemosa-cimicifuga-racemosa-se-comporta-como-un-ligando-competitivo-mixto-y-agonista-parcial-en-el-receptor-opiaceo-%ce%bc-humano","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=45278","title":{"rendered":"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria &#8211; HERBOLOGIA: \u00abCohosh negro (Actaea racemosa, Cimicifuga racemosa) se comporta como un ligando competitivo mixto y agonista parcial en el receptor opi\u00e1ceo \u03bc humano\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-66fIpCGXX60\/X-Uamt99N8I\/AAAAAAAAhWU\/HIwyyuvGEGoxmo-z5Kh4CM-3U86tV4LpACLcBGAsYHQ\/s950\/Journal_agricultural%2Band%2Bfood%2Bchemistry3.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-66fIpCGXX60\/X-Uamt99N8I\/AAAAAAAAhWU\/HIwyyuvGEGoxmo-z5Kh4CM-3U86tV4LpACLcBGAsYHQ\/s320\/Journal_agricultural%2Band%2Bfood%2Bchemistry3.jpg\" height=\"320\" border=\"0\" data-original-height=\"950\" data-original-width=\"714\" \/><\/a>Rhyu, M. R., Lu, J., Webster, D. E., Fabricant, D. S., Farnsworth, N. R., &amp; Wang, Z. J. (2006). <a href=\"https:\/\/www.ncbi.nlm.nih.gov\/pmc\/articles\/PMC2547488\/\">Black cohosh (Actaea racemosa, Cimicifuga racemosa) behaves as a mixed competitive ligand and partial agonist at the human \u03bc opiate receptor<\/a>.<i>\u00a0Journal of agricultural and food chemistry<\/i>, 54(26), 9852-9857.<\/p>\n<p>El cohosh negro es un suplemento diet\u00e9tico bot\u00e1nico de uso com\u00fan para el tratamiento de las molestias climat\u00e9ricas. Dado que el sistema de opi\u00e1ceos en el cerebro est\u00e1 \u00edntimamente asociado con el estado de \u00e1nimo, la temperatura y los niveles hormonales sexuales, investigamos la actividad de los extractos de cohosh negro en el receptor opi\u00e1ceo \u03bc humano (hMOR) expresado en c\u00e9lulas de ovario de h\u00e1mster chino.<\/p>\n<p>Los extractos de cohosh negro 100% metanol, 75% etanol y 40% 2-propanol desplazaron eficazmente la uni\u00f3n espec\u00edfica de [3H] DAMGO a hMOR. Estudios adicionales del extracto de etanol usado cl\u00ednicamente indicaron que el cohosh negro actu\u00f3 como un ligando competitivo mixto, desplazando el 77 \u00b1 4% de [3H] DAMGO a hMOR (Ki = 62,9 \u00b5g \/ ml). Usando el ensayo de [35S] GTP\u03b3S, se encontr\u00f3 que la acci\u00f3n del cohosh negro era consistente con un agonista, con una CE50 de 68,8 \u00b1 7,7 \u00b5g \/ ml.<\/p>\n<p>CONCLUSION: Estos resultados demuestran por primera vez que el cohosh negro contiene principios activos que activan el hMOR, lo que respalda su funci\u00f3n beneficiosa para aliviar los s\u00edntomas de la menopausia.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Rhyu, M. R., Lu, J., Webster, D. E., Fabricant, D. S., Farnsworth, N. R., &amp; Wang, Z. J. (2006). Black cohosh (Actaea racemosa, Cimicifuga racemosa) behaves as a mixed competitive ligand and partial agonist at the human \u03bc opiate receptor.\u00a0Journal of agricultural and food chemistry, 54(26), 9852-9857. El cohosh negro es un suplemento diet\u00e9tico bot\u00e1nico [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[5],"tags":[],"class_list":["post-45278","post","type-post","status-publish","format-standard","hentry","category-naturopatia-fitocomplementaria-herbologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;Cohosh negro (Actaea racemosa, Cimicifuga racemosa) se comporta como un ligando competitivo mixto y agonista parcial en el receptor opi\u00e1ceo \u03bc humano&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: &quot;Cohosh negro (Actaea racemosa, Cimicifuga racemosa) se comporta como un ligando competitivo mixto y agonista parcial en el receptor opi\u00e1ceo \u03bc humano&quot; -\" \/>\n<meta property=\"og:description\" content=\"Rhyu, M. R., Lu, J., Webster, D. E., Fabricant, D. S., Farnsworth, N. R., &amp; Wang, Z. J. (2006). Black cohosh (Actaea racemosa, Cimicifuga racemosa) behaves as a mixed competitive ligand and partial agonist at the human \u03bc opiate receptor.\u00a0Journal of agricultural and food chemistry, 54(26), 9852-9857. El cohosh negro es un suplemento diet\u00e9tico bot\u00e1nico [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\" \/>\n<meta property=\"article:published_time\" content=\"2020-12-23T00:30:18+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2020-12-25T09:39:57+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-66fIpCGXX60\/X-Uamt99N8I\/AAAAAAAAhWU\/HIwyyuvGEGoxmo-z5Kh4CM-3U86tV4LpACLcBGAsYHQ\/s320\/Journal_agricultural%2Band%2Bfood%2Bchemistry3.jpg\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" content=\"Tiempo de lectura\" \/>\n\t<meta name=\"twitter:data2\" content=\"1 minuto\" \/>\n<script type=\"application\/ld+json\" class=\"yoast-schema-graph\">{\"@context\":\"https:\/\/schema.org\",\"@graph\":[{\"@type\":\"Article\",\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278#article\",\"isPartOf\":{\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\"},\"author\":{\"name\":\"admin\",\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/#\/schema\/person\/432852c9ed996fc42e869a813ecbffd7\"},\"headline\":\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria &#8211; HERBOLOGIA: \u00abCohosh negro (Actaea racemosa, Cimicifuga racemosa) se comporta como un ligando competitivo mixto y agonista parcial en el receptor opi\u00e1ceo \u03bc humano\u00bb\",\"datePublished\":\"2020-12-23T00:30:18+00:00\",\"dateModified\":\"2020-12-25T09:39:57+00:00\",\"mainEntityOfPage\":{\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\"},\"wordCount\":269,\"commentCount\":0,\"publisher\":{\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/#organization\"},\"articleSection\":[\"Naturopat\u00eda Fitocomplementaria HERBOLOG\u00cdA\"],\"inLanguage\":\"es\",\"potentialAction\":[{\"@type\":\"CommentAction\",\"name\":\"Comment\",\"target\":[\"https:\/\/rina.naturopatiadigital.eu\/?p=45278#respond\"]}]},{\"@type\":\"WebPage\",\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\",\"url\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\",\"name\":\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria - HERBOLOGIA: \\\"Cohosh negro (Actaea racemosa, Cimicifuga racemosa) se comporta como un ligando competitivo mixto y agonista parcial en el receptor opi\u00e1ceo \u03bc humano\\\" -\",\"isPartOf\":{\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/#website\"},\"datePublished\":\"2020-12-23T00:30:18+00:00\",\"dateModified\":\"2020-12-25T09:39:57+00:00\",\"breadcrumb\":{\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278#breadcrumb\"},\"inLanguage\":\"es\",\"potentialAction\":[{\"@type\":\"ReadAction\",\"target\":[\"https:\/\/rina.naturopatiadigital.eu\/?p=45278\"]}]},{\"@type\":\"BreadcrumbList\",\"@id\":\"https:\/\/rina.naturopatiadigital.eu\/?p=45278#breadcrumb\",\"itemListElement\":[{\"@type\":\"ListItem\",\"position\":1,\"name\":\"Home\",\"item\":\"https:\/\/rina.naturopatiadigital.eu\/\"},{\"@type\":\"ListItem\",\"position\":2,\"name\":\"\u00c1rea de conocimiento: Tecnolog\u00eda Naturop\u00e1tica o Naturopat\u00eda Aplicada: M\u00f3dulo: Naturopat\u00eda Fitocomplementaria &#8211; 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