{"id":45341,"date":"2020-12-26T07:30:16","date_gmt":"2020-12-26T06:30:16","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=45341"},"modified":"2020-12-26T20:49:44","modified_gmt":"2020-12-26T19:49:44","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-tuyona-inhibe-la-metastasis-pulmonar-inducida-por-celulas-de-melanoma-b16f-10-en-ratones-c57bl-6","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=45341","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abTuyona inhibe la met\u00e1stasis pulmonar inducida por c\u00e9lulas de melanoma B16F-10 en ratones C57BL \/ 6\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-tcLUQhy71B8\/X-eTJOkJh6I\/AAAAAAAAhbY\/FyktQdFDwGgmzxV-xsabPkm28rMpdeoUACLcBGAsYHQ\/s375\/Canadian_journal%2Bof%2Bphysiology%2Band%2Bpharmacology.jpg\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-tcLUQhy71B8\/X-eTJOkJh6I\/AAAAAAAAhbY\/FyktQdFDwGgmzxV-xsabPkm28rMpdeoUACLcBGAsYHQ\/s320\/Canadian_journal%2Bof%2Bphysiology%2Band%2Bpharmacology.jpg\" height=\"320\" border=\"0\" data-original-height=\"375\" data-original-width=\"290\" \/><\/a>Siveen, K. S., &amp; Kuttan, G. (2011). <a href=\"https:\/\/www.researchgate.net\/profile\/Kodappully-Siveen\/publication\/51637384_Thujone_inhibits_lung_metastasis_induced_by_B16F-10_melanoma_cells_in_C57BL6_mice\/links\/0a85e52d7905863f00000000\/Thujone-inhibits-lung-metastasis-induced-by-B16F-10-melanoma-cells-in-C57BL-6-mice.pdf\">Thujone inhibits lung metastasis induced by B16F-10 melanoma cells in C57BL\/6 mice<\/a>.<i>\u00a0Canadian journal of physiology and pharmacology<\/i>, 89(10), 691-703.<\/p>\n<p>OBJETIVO: Se evalu\u00f3 el potencial antimetast\u00e1sico de la tuyona, un monoterpeno natural.<\/p>\n<p>METODOLOGIA: Se indujo met\u00e1stasis en ratones C57BL \/ 6 inyectando c\u00e9lulas de melanoma B16F-10 altamente metast\u00e1sicas a trav\u00e9s de la vena lateral de la cola.<\/p>\n<p>RESULTADOS: La administraci\u00f3n de tuyona (1 mg \u00b7 (kg de peso corporal) (- 1)), profil\u00e1cticamente y simult\u00e1neamente con la inducci\u00f3n tumoral, inhibi\u00f3 la formaci\u00f3n de n\u00f3dulos tumorales en los pulmones en un 59,45% y 57,54%, respectivamente, con un aumento en la tasa de supervivencia (33,67 % y 32,16%) de los animales portadores de tumores metast\u00e1sicos. Estos resultados se correlacionaron con par\u00e1metros bioqu\u00edmicos como el contenido de hidroxiprolina, hexosamina y \u00e1cido ur\u00f3nico de col\u00e1geno pulmonar, niveles s\u00e9ricos de \u00e1cido si\u00e1lico y \u03b3-glutamil transpeptidasa y an\u00e1lisis histopatol\u00f3gico. El tratamiento con tuyona regul\u00f3 negativamente la producci\u00f3n de citocinas proinflamatorias como el factor de necrosis tumoral \u03b1, la interleucina (IL) -1\u03b2, la IL-6 y el factor estimulante de colonias de granulocitos y monocitos. La administraci\u00f3n de tujona regul\u00f3 negativamente la expresi\u00f3n de metaloproteinasa de matriz (MMP) -2, MMP-9, quinasa regulada por se\u00f1al extracelular (ERK) -1, ERK-2 y factor de crecimiento endotelial vascular (VEGF) y tambi\u00e9n regul\u00f3 positivamente la expresi\u00f3n de nm-23 , inhibidor tisular de metaloproteinasa (TIMP) -1 y TIMP-2 en el tejido pulmonar de animales inducidos por met\u00e1stasis. El tratamiento con tuyona inhibi\u00f3 la actividad de MMP-2 y MMP-9 en el an\u00e1lisis zimogr\u00e1fico de gelatina. El tratamiento con tuyona inhibi\u00f3 significativamente la invasi\u00f3n de c\u00e9lulas de melanoma B16F-10 a trav\u00e9s de la matriz de col\u00e1geno en una c\u00e1mara de Boyden. La tuyona tambi\u00e9n inhibi\u00f3 la adhesi\u00f3n de las c\u00e9lulas tumorales a los pocillos de la placa de microtiro recubiertos de col\u00e1geno y la migraci\u00f3n de c\u00e9lulas de melanoma B16F-10 a trav\u00e9s de un filtro de policarbonato in vitro.<\/p>\n<p>CONCLUSION: Estos resultados indican que la tuyona puede inhibir la met\u00e1stasis pulmonar de c\u00e9lulas B16F-10 mediante la inhibici\u00f3n de la proliferaci\u00f3n, adhesi\u00f3n e invasi\u00f3n de c\u00e9lulas tumorales, as\u00ed como regulando la expresi\u00f3n de MMP, VEGF, ERK-1, ERK-2, TIMP, nm23, y niveles de citocinas proinflamatorias e IL-2 en animales metast\u00e1sicos.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Siveen, K. S., &amp; Kuttan, G. (2011). Thujone inhibits lung metastasis induced by B16F-10 melanoma cells in C57BL\/6 mice.\u00a0Canadian journal of physiology and pharmacology, 89(10), 691-703. OBJETIVO: Se evalu\u00f3 el potencial antimetast\u00e1sico de la tuyona, un monoterpeno natural. METODOLOGIA: Se indujo met\u00e1stasis en ratones C57BL \/ 6 inyectando c\u00e9lulas de melanoma B16F-10 altamente metast\u00e1sicas a [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-45341","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Tuyona inhibe la met\u00e1stasis pulmonar inducida por c\u00e9lulas de melanoma B16F-10 en ratones C57BL \/ 6&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=45341\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Tuyona inhibe la met\u00e1stasis pulmonar inducida por c\u00e9lulas de melanoma B16F-10 en ratones C57BL \/ 6&quot; -\" \/>\n<meta property=\"og:description\" content=\"Siveen, K. S., &amp; Kuttan, G. (2011). Thujone inhibits lung metastasis induced by B16F-10 melanoma cells in C57BL\/6 mice.\u00a0Canadian journal of physiology and pharmacology, 89(10), 691-703. OBJETIVO: Se evalu\u00f3 el potencial antimetast\u00e1sico de la tuyona, un monoterpeno natural. METODOLOGIA: Se indujo met\u00e1stasis en ratones C57BL \/ 6 inyectando c\u00e9lulas de melanoma B16F-10 altamente metast\u00e1sicas a [&hellip;]\" \/>\n<meta property=\"og:url\" content=\"https:\/\/rina.naturopatiadigital.eu\/?p=45341\" \/>\n<meta property=\"article:published_time\" content=\"2020-12-26T06:30:16+00:00\" \/>\n<meta property=\"article:modified_time\" content=\"2020-12-26T19:49:44+00:00\" \/>\n<meta property=\"og:image\" content=\"https:\/\/1.bp.blogspot.com\/-tcLUQhy71B8\/X-eTJOkJh6I\/AAAAAAAAhbY\/FyktQdFDwGgmzxV-xsabPkm28rMpdeoUACLcBGAsYHQ\/s320\/Canadian_journal%2Bof%2Bphysiology%2Band%2Bpharmacology.jpg\" \/>\n<meta name=\"author\" content=\"admin\" \/>\n<meta name=\"twitter:card\" content=\"summary_large_image\" \/>\n<meta name=\"twitter:label1\" content=\"Escrito por\" \/>\n\t<meta name=\"twitter:data1\" content=\"admin\" \/>\n\t<meta name=\"twitter:label2\" content=\"Tiempo de lectura\" \/>\n\t<meta name=\"twitter:data2\" content=\"2 minutos\" \/>\n<script 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