{"id":45552,"date":"2021-01-27T05:30:25","date_gmt":"2021-01-27T04:30:25","guid":{"rendered":"https:\/\/rina.naturopatiadigital.eu\/?p=45552"},"modified":"2021-01-31T20:23:46","modified_gmt":"2021-01-31T19:23:46","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-el-barakol-un-ansiolitico-natural-inhibe-la-liberacion-de-dopamina-estriatal-pero-no-la-captacion-in-vitro","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=45552","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abEl barakol, un ansiol\u00edtico natural, inhibe la liberaci\u00f3n de dopamina estriatal pero no la captaci\u00f3n in vitro\u00bb"},"content":{"rendered":"<p><a href=\"https:\/\/1.bp.blogspot.com\/-3yfBVXIZIkk\/YBcCwnbgyXI\/AAAAAAAAhrI\/qczL9zwx3zwA_1ARcKOLsQVnGAxfHk6wACLcBGAsYHQ\/s160\/European_journal%2Bof%2Bpharmacology.gif\"><img decoding=\"async\" class=\"alignleft\" src=\"https:\/\/1.bp.blogspot.com\/-3yfBVXIZIkk\/YBcCwnbgyXI\/AAAAAAAAhrI\/qczL9zwx3zwA_1ARcKOLsQVnGAxfHk6wACLcBGAsYHQ\/s0\/European_journal%2Bof%2Bpharmacology.gif\" border=\"0\" data-original-height=\"160\" data-original-width=\"120\" \/><\/a>Thongsaard, W., Pongsakorn, S., Sudsuang, R., Bennett, G. W., Kendall, D. A., &amp; Marsden, C. A. (1997). <a href=\"https:\/\/www.sciencedirect.com\/science\/article\/abs\/pii\/S0014299996008503\">Barakol, a natural anxiolytic, inhibits striatal dopamine release but not uptake in vitro<\/a>. <i>European journal of pharmacology<\/i>, 319(2-3), 157-164.<\/p>\n<p>OBJETIVO \/ METODO:: El presente estudio investig\u00f3 los efectos del barakol sobre la liberaci\u00f3n in vitro de dopamina end\u00f3gena y radiomarcada de cortes estriatales de rata en comparaci\u00f3n con los agonistas del receptor de dopamina, el diclorhidrato de quinelorano (1 \u03bcM) y el metanosulfonato de pergolida (100 \u03bcM), y el antagonista del receptor de dopamina, S (-) &#8211; clorhidrato de eticloprida (10 \u03bcM) utilizando un m\u00e9todo de semi-superfusi\u00f3n y cromatograf\u00eda l\u00edquida de alta resoluci\u00f3n con medici\u00f3n de detector electroqu\u00edmico de dopamina end\u00f3gena.<\/p>\n<p>RESULTADOS: El barakol (1, 10 y 100 \u00b5M) redujo la liberaci\u00f3n de dopamina end\u00f3gena estimulada por K + al igual que los agonistas del receptor de dopamina D2, pero no tuvo ning\u00fan efecto sobre la liberaci\u00f3n de dopamina [3H]. La inhibici\u00f3n de barakol (10 \u00b5M) sobre la liberaci\u00f3n de dopamina end\u00f3gena estimulada por K + fue antagonizada por un antagonista del receptor de dopamina D2, eticloprida. El barakol (0,1 nM \u2013 10 \u00b5M) no tuvo ning\u00fan efecto sobre la captaci\u00f3n de [3H] dopamina, excepto a la concentraci\u00f3n m\u00e1s alta (100 \u00b5M) cuando se observ\u00f3 inhibici\u00f3n.<\/p>\n<p>CONCLUSION: Los resultados indican que el barakol podr\u00eda actuar como agonista de la dopamina para inhibir la liberaci\u00f3n de dopamina end\u00f3gena sin un cambio en la captaci\u00f3n de dopamina.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Thongsaard, W., Pongsakorn, S., Sudsuang, R., Bennett, G. W., Kendall, D. A., &amp; Marsden, C. A. (1997). Barakol, a natural anxiolytic, inhibits striatal dopamine release but not uptake in vitro. European journal of pharmacology, 319(2-3), 157-164. OBJETIVO \/ METODO:: El presente estudio investig\u00f3 los efectos del barakol sobre la liberaci\u00f3n in vitro de dopamina end\u00f3gena [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[5],"tags":[],"class_list":["post-45552","post","type-post","status-publish","format-standard","hentry","category-naturopatia-fitocomplementaria-herbologia"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El barakol, un ansiol\u00edtico natural, inhibe la liberaci\u00f3n de dopamina estriatal pero no la captaci\u00f3n in vitro&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=45552\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;El barakol, un ansiol\u00edtico natural, inhibe la liberaci\u00f3n de dopamina estriatal pero no la captaci\u00f3n in vitro&quot; -\" \/>\n<meta property=\"og:description\" content=\"Thongsaard, W., Pongsakorn, S., Sudsuang, R., Bennett, G. 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