{"id":46380,"date":"2024-07-23T15:00:16","date_gmt":"2024-07-23T13:00:16","guid":{"rendered":"https:\/\/RevistaEspa\u00f1olaNaturopatia.naturopatiadigital.eu\/?p=46380"},"modified":"2024-07-23T15:00:47","modified_gmt":"2024-07-23T13:00:47","slug":"area-de-conocimiento-naturopatia-experimental-sustancias-bioactivas-actividad-antitumoral-de-la-arctigenina-en-la-linea-celular-t24-del-cancer-de-vejiga-mediante-la-induccion-de-la-detencion-del","status":"publish","type":"post","link":"https:\/\/rina.naturopatiadigital.eu\/?p=46380","title":{"rendered":"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: \u00abActividad antitumoral de la arctigenina en la l\u00ednea celular T24 del c\u00e1ncer de vejiga mediante la inducci\u00f3n de la detenci\u00f3n del ciclo celular y la apoptosis\u00bb"},"content":{"rendered":"<p><img decoding=\"async\" src=\"https:\/\/i1.rgstatic.net\/publication\/332876135_The_Anatomical_Record_Advances_in_Integrative_Anatomy_and_Evolutionary_Biology_A_R_C_elebrating_OVER_100_YEARS_of_E_xcellence_in_ANATOMICAL_PUBLICATION\/links\/5cd00383a6fdccc9dd902584\/largepreview.png\" alt=\"PDF) The Anatomical Record Advances in Integrative Anatomy and Evolutionary Biology A R C elebrating OVER 100 YEARS of E xcellence in ANATOMICAL PUBLICATION\" \/><img decoding=\"async\" src=\"https:\/\/i1.rgstatic.net\/publication\/332876135_The_Anatomical_Record_Advances_in_Integrative_Anatomy_and_Evolutionary_Biology_A_R_C_elebrating_OVER_100_YEARS_of_E_xcellence_in_ANATOMICAL_PUBLICATION\/links\/5cd00383a6fdccc9dd902584\/largepreview.png\" alt=\"PDF) The Anatomical Record Advances in Integrative Anatomy and Evolutionary Biology A R C elebrating OVER 100 YEARS of E xcellence in ANATOMICAL PUBLICATION\" \/><img decoding=\"async\" src=\"https:\/\/i1.rgstatic.net\/publication\/332876135_The_Anatomical_Record_Advances_in_Integrative_Anatomy_and_Evolutionary_Biology_A_R_C_elebrating_OVER_100_YEARS_of_E_xcellence_in_ANATOMICAL_PUBLICATION\/links\/5cd00383a6fdccc9dd902584\/largepreview.png\" alt=\"PDF) The Anatomical Record Advances in Integrative Anatomy and Evolutionary Biology A R C elebrating OVER 100 YEARS of E xcellence in ANATOMICAL PUBLICATION\" \/><img fetchpriority=\"high\" decoding=\"async\" class=\"alignleft\" src=\"https:\/\/anatomypubs.onlinelibrary.wiley.com\/cms\/asset\/2b53170e-8eac-4d01-8ec8-2a6e00567422\/ar.v304.4.cover.gif\" width=\"202\" height=\"266\" \/>Yang, S., Ma, J., Xiao, J., Lv, X., Li, X., Yang, H., &#8230; &amp; Zhang, Y. (2012). <a href=\"https:\/\/anatomypubs.onlinelibrary.wiley.com\/doi\/full\/10.1002\/ar.22497\">Arctigenin anti\u2010tumor activity in bladder cancer T24 cell line through induction of cell\u2010cycle arrest and apoptosis.<\/a>\u00a0<i>The Anatomical Record: Advances in Integrative Anatomy and Evolutionary Biology<\/i>,\u00a0<i>295<\/i>(8), 1260-1266.<\/p>\n<p>CONTEXTO. El c\u00e1ncer de vejiga es la neoplasia m\u00e1s com\u00fan en el sistema urinario.<\/p>\n<p>OBJETIVO. Este estudio eval\u00faa la actividad antitumoral de la arctigenina en c\u00e9lulas T24 de c\u00e1ncer de vejiga humano in vitro y los eventos moleculares subyacentes.<\/p>\n<p>METODO. El an\u00e1lisis de citometr\u00eda de flujo se utiliz\u00f3 para detectar la distribuci\u00f3n del ciclo celular y la apoptosis. Se utiliz\u00f3 Western blotting para detectar cambios en la expresi\u00f3n de prote\u00ednas.<\/p>\n<p>RESULTADOS. Los datos mostraron que el tratamiento con arctigenina redujo la viabilidad de las c\u00e9lulas T24 de c\u00e1ncer de vejiga de manera dependiente de la dosis y el tiempo despu\u00e9s del tratamiento con arctigenina (10, 20, 40, 80 y 100 \u03bcmol\/L) durante 24 horas y 48 horas. El tratamiento con arctigenina detuvo claramente las c\u00e9lulas tumorales en la fase G1 del ciclo celular. La apoptosis se detect\u00f3 mediante tinci\u00f3n de Hoechst y citometr\u00eda de flujo despu\u00e9s de la tinci\u00f3n doble con Annexin-V-FITC\/PI. Las c\u00e9lulas apopt\u00f3ticas tempranas y tard\u00edas representaron el 2,32-7,01% y el 3,07-7,35%, respectivamente. A nivel molecular, el tratamiento con arctigenina disminuy\u00f3 la expresi\u00f3n de ciclina D1, mientras que los niveles de expresi\u00f3n de CDK4 y CDK6 no se vieron afectados. Adem\u00e1s, la arctigenina alter\u00f3 selectivamente la fosforilaci\u00f3n de los miembros de la superfamilia MAPK, disminuyendo la fosforilaci\u00f3n de ERK1\/2 y activando la fosforilaci\u00f3n de p38 significativamente de manera dependiente de la dosis.<\/p>\n<p>CONCLUSIONES. Estos resultados sugieren que la arctigenina puede inhibir la viabilidad celular e inducir la apoptosis mediante la activaci\u00f3n directa de la v\u00eda mitocondrial, y la v\u00eda de la prote\u00edna quinasa activada por mit\u00f3geno puede desempe\u00f1ar un papel importante en el efecto antitumoral de la arctigenina. Los datos del estudio actual demuestran la utilidad de la arctigenina en las c\u00e9lulas T24 del c\u00e1ncer de vejiga, que deben evaluarse m\u00e1s a fondo in vivo antes de traducirse en ensayos cl\u00ednicos para la quimioprevenci\u00f3n del c\u00e1ncer de vejiga.<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Yang, S., Ma, J., Xiao, J., Lv, X., Li, X., Yang, H., &#8230; &amp; Zhang, Y. (2012). Arctigenin anti\u2010tumor activity in bladder cancer T24 cell line through induction of cell\u2010cycle arrest and apoptosis.\u00a0The Anatomical Record: Advances in Integrative Anatomy and Evolutionary Biology,\u00a0295(8), 1260-1266. CONTEXTO. El c\u00e1ncer de vejiga es la neoplasia m\u00e1s com\u00fan en el [&hellip;]<\/p>\n","protected":false},"author":1,"featured_media":0,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[8],"tags":[],"class_list":["post-46380","post","type-post","status-publish","format-standard","hentry","category-sustancias-bioactivas"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v21.8 - https:\/\/yoast.com\/wordpress\/plugins\/seo\/ -->\n<title>\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Actividad antitumoral de la arctigenina en la l\u00ednea celular T24 del c\u00e1ncer de vejiga mediante la inducci\u00f3n de la detenci\u00f3n del ciclo celular y la apoptosis&quot; -<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/rina.naturopatiadigital.eu\/?p=46380\" \/>\n<meta property=\"og:locale\" content=\"es_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"\u00c1rea de conocimiento: Naturopat\u00eda Experimental: Sustancias Bioactivas: &quot;Actividad antitumoral de la arctigenina en la l\u00ednea celular T24 del c\u00e1ncer de vejiga mediante la inducci\u00f3n de la detenci\u00f3n del ciclo celular y la apoptosis&quot; -\" \/>\n<meta property=\"og:description\" content=\"Yang, S., Ma, J., Xiao, J., Lv, X., Li, X., Yang, H., &#8230; &amp; Zhang, Y. 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